Target Names are taken from UniProtKB. To view the associated UniProt page, click on the UniProt ID. When we have data for a given Target in multiple species or for mutants of a given Target, we provide a header row (upper case, bold font) with all of the data followed by a separate for each species or variant of the Target.
Target Name
Organism
Affinity Links
Articles
UniProts
Files
Human
Human
Human
Human
Human
Spiny starfish
Human
IC50: 1
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3 O95067 P06493 P14635 Q8WWL7
Human
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3/cAMP-dependent protein kinase O95067 P06493 P14635 Q8WWL7 Q95J97
Rabbit
IC50: 1
Human
GAG-POL POLYPROTEIN P03354 P03359 P03366 P03367 P03369 P04584 P04585 P05959 P06633 P0C6F2 P12497 P24740 Q04095 Q9QBY3
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 6
Human immunodeficiency virus type 1
Ki: 1
Dimer of Gag-Pol polyprotein [489-587,K509R,V521I,L522F,M525I,I543V,L552P,A560V,V571A,I573V,L579M] P04585
Human immunodeficiency virus type 1
Ki: 4
Human immunodeficiency virus type 1
Ki: 4
Human immunodeficiency virus type 1
Ki: 4
Human immunodeficiency virus type 1
Ki: 4
Dimer of Gag-Pol polyprotein [489-587,K509R,V521I,L522F,M525I,M535I,I543V,L552P,A560V,V571A,I573V,L579M] P04585
Human immunodeficiency virus type 1
Ki: 4
Dimer of Gag-Pol polyprotein [489-587,K509R,V521I,L522F,M525I,M535I,L552P,A560V,V571A,I573V,L579M] P04585
Human immunodeficiency virus type 1
Ki: 4
Human immunodeficiency virus type 1
Ki: 4
Dimer of Gag-Pol polyprotein [489-587,L499I,L508Q,K509R,E524D,M525I,S526N,M535I,I539V,I543V,I551V,L552P,A560V,V571A,L579M] P04585
Human immunodeficiency virus type 1
Ki: 6
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 6
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,M525I,N526D,M535I,R546K,L552P,A560V,G562S,I573V,L579M,I582L] P12497
Human immunodeficiency virus type 1
IC50: 27
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,M535I,I543V,Q547E,L552P,I553V,V566I,V571F,I573V,L579M,I582L] P12497
Human immunodeficiency virus type 1
IC50: 15
Dimer of Gag-Pol polyprotein [489-587,Q496K,L499I,N526S,R530K,M535I,I543V,I551V,L552P,A560V,V566I,V571A,L579M,I582L] P12497
Human immunodeficiency virus type 1
IC50: 11
Human immunodeficiency virus type 1
IC50: 73
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 62
Human immunodeficiency virus type 1
Ki: 19
Human immunodeficiency virus type 1
Ki: 19
Human immunodeficiency virus type 1
Ki: 19
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Ki: 2
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 8
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus 2
Human immunodeficiency virus type 1
IC50: 3
Human immunodeficiency virus
Ki: 10
Human immunodeficiency virus
Ki: 10
Human immunodeficiency virus
Ki: 9
Gag-Pol polyprotein [484-582,I497V,V499I,E519D,R541K,D544E,Q553K,A555V,G557S,I568V,L574M,L573M] Q9QBY3
Human immunodeficiency virus
Ki: 10
Gag-Pol polyprotein [484-582,Q491K,I494L,I497V,V499I,E519D,I534V,R541K,D544E,Q553K,A555V,L573M] Q9QBY3
Human immunodeficiency virus
Ki: 11
Human immunodeficiency virus
Ki: 11
Gag-Pol polyprotein [484-582,Q491K,I497V,V499I,E519D,G532V,I538V,R541K,D544E,L547P,Q553K,V566A,L573M] Q9QBY3
Human immunodeficiency virus
Ki: 11
Gag-Pol polyprotein [484-582,Q491K,I497V,V499I,E519D,R541K,D544E,L547P,Q553K,A555V,G557S,I568V,L573M,L574M] Q9QBY3
Human immunodeficiency virus
Ki: 11
Human immunodeficiency virus
Human immunodeficiency virus type 1
EC50: 83
Human immunodeficiency virus type 1
Gag-Pol polyprotein [489-892,N526H,R530K,V566I,I582L,V648I,Q690K,I723V,C750S,T788A,Q795E,T874A,V881I,P882Q] P12497
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus type 1
IC50: 84
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
IC50: 42
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
IC50: 1143
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
IC50: 181
Human immunodeficiency virus type 1
IC50: 9
Human immunodeficiency virus type 1
IC50: 11
Human immunodeficiency virus type 1
IC50: 10
Human immunodeficiency virus type 1
IC50: 10
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
IC50: 9
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
Human immunodeficiency virus type 1
IC50: 18
Gag-Pol polyprotein [600-1028,D666N,K669R,T814F,K818Q,C879S]/[600-1151,D666N,K669R,T814F,K818Q,C879S] P03366
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 43
Gag-Pol polyprotein [600-1159,Y780C]/Imidazoleglycerol-phosphate dehydratase [600-1029,Y780C] P03366 P06633
Human immunodeficiency virus type 1
IC50: 3
Human immunodeficiency virus 2
IC50: 5
Human immunodeficiency virus type 1
EC50: 6
Rat
Human
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1 O14764 P08219 P08220 P14867 P18505 P18506 P18507 P18508 P22723 P28472 P47870 P62812 P62813 P63079 P63138 Q8N1C3
Human
Human
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-200],P14867[176-456] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,A118C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,D95C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,F116C] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,L179C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,M169C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R171C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R183C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R233C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T120C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T165C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T181C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-3 [26-473]/gamma-2 [40-467] P14867 P18507 P28472
Human
Ki: 8
Gamma-aminobutyric acid receptor subunit alpha-1 [A160C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [D97C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [F99C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G157C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G200C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S204C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S205C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T162C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T206C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V211C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [Y209C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Human
Human
Ki: 112
Human
Rat
Rat
EC50: 2
Human
Rat
Rat
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-2 P18506 P18507 P18508 P23576 P28472 P47869 P47870 P63079 P63138 Q8N1C3
Human
Human
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47869 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P47869
Human
Ki: 8
Human
Ki: 273
Rat
Ki: 25
Human
Rat
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-3 P18507 P18508 P20236 P28472 P34903 P47870 P63079 P63138
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-2 [26-512]/gamma-2 [40-467] P18507 P34903 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P34903
Human
Ki: 7
Rat
Ki: 26
Human
Human
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-4 O14764 P18505 P18506 P18507 P18508 P28471 P28472 P47870 P48169 P63079
Human
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 P48169
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P48169
Human
Ki: 4
Human
Human
EC50: 1
Human
EC50: 18
Rat
Human
EC50: 12
Rat
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-5 P18507 P18508 P19969 P28472 P31644 P47870 P63079 Q8N1C3
Human
Human
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-2 [26-512]/gamma-2 [40-467] P18507 P31644 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P31644
Human
Ki: 11
Human
Ki: 190
Human
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-6 P18506 P18507 P18508 P28472 P30191 P47870 P63079 P63138 Q16445
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 Q16445
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 Q16445
Human
Ki: 7
Rat
Human
Ki: 20
Rat
Rat
Rat
IC50: 10
Human
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-1 O14764 P08219 P08220 P14867 P15431 P18505 P18507 P47870 P48169
Human
Human
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-2 O14764 P14867 P18505 P18506 P18507 P18508 P20236 P23576 P30191 P31644 P34903 P47869 P47870 P48169 P62813 P63138 Q16445 Q8N1C3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-200],P14867[176-456] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,A118C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,D95C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,F116C] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,L179C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,M169C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R171C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R183C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R233C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T120C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T165C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T181C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [A160C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [D97C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [F99C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G157C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G200C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S204C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S205C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T162C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T206C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V211C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [Y209C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Human
Human
Ki: 112
Human
Rat
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47869 P47870
Human
Ki: 3
Human
Ki: 273
Rat
Ki: 25
Human
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-2 [26-512]/gamma-2 [40-467] P18507 P34903 P47870
Human
Ki: 3
Rat
Ki: 26
Human
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 P48169
Human
Ki: 3
Human
EC50: 1
Human
EC50: 18
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-2 [26-512]/gamma-2 [40-467] P18507 P31644 P47870
Human
Ki: 3
Human
Ki: 190
Human
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 Q16445
Human
Ki: 3
Rat
Human
Ki: 20
Rat
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-3 O14764 P14867 P18506 P18507 P18508 P19969 P20236 P22723 P23576 P28471 P28472 P30191 P31644 P34903 P47869 P48169 P62813 P63079 Q16445
Human
Human
Human
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-3 [26-473]/gamma-2 [40-467] P14867 P18507 P28472
Human
Ki: 8
Rat
EC50: 2
Human
Rat
Rat
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P47869
Human
Ki: 8
Rat
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P34903
Human
Ki: 7
Human
Rat
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P48169
Human
Ki: 4
Rat
Human
EC50: 12
Rat
Rat
IC50: 1
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P31644
Human
Ki: 11
Rat
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 Q16445
Human
Ki: 7
Rat
Rat
IC50: 10
Human
Rat
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT DELTA O14764 P14867 P18505 P18506 P23576 P28471 P28472 P30191 P47870 P48169 P62813 P63079 P63138
Human
Rat
EC50: 2
Human
Human
EC50: 1
Human
EC50: 12
Rat
Rat
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT GAMMA-2 P14867 P18505 P18507 P18508 P19969 P20236 P22723 P23576 P28471 P28472 P30191 P31644 P34903 P47869 P47870 P48169 P62813 P63079 P63138 Q16445
Human
Human
Human
Human
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-200],P14867[176-456] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,A118C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,D95C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,F116C] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,L179C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,M169C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R171C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R183C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R224C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,R233C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T120C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T165C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,T181C] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-3 [26-473]/gamma-2 [40-467] P14867 P18507 P28472
Human
Ki: 8
Gamma-aminobutyric acid receptor subunit alpha-1 [A160C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [D97C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Gamma-aminobutyric acid receptor subunit alpha-1 [F99C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G157C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [G200C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S204C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [S205C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T162C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [T206C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V202C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [V211C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-1 [Y209C]/beta-2 [26-512]/gamma-2 [40-467] P14867 P18507 P47870
Human
Other: 1
Human
Rat
Human
Rat
Rat
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47869 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-2 [29-451]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P47869
Human
Ki: 8
Rat
Ki: 25
Human
Rat
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-2 [26-512]/gamma-2 [40-467] P18507 P34903 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P34903
Human
Ki: 7
Rat
Ki: 26
Human
Human
Rat
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 P48169
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-4 [36-554]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P48169
Human
Ki: 4
Human
EC50: 18
Rat
IC50: 1
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-2 [26-512]/gamma-2 [40-467] P18507 P31644 P47870
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-5 [32-462]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 P31644
Human
Ki: 11
Human
Rat
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-2 [26-512]/gamma-2 [40-467] P18507 P47870 Q16445
Human
Ki: 3
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-3 [26-473]/gamma-2 [40-467] P18507 P28472 Q16445
Human
Ki: 7
Human
Ki: 20
Rat
Human
Rat
Human
Rat
Human
Rat
Human
Human
Gamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2 P49768 P49810 Q8WW43 Q92542 Q96BI3 Q9NZ42
Human
IC50: 558
GASTRIN/CHOLECYSTOKININ TYPE B RECEPTOR H0VZC5 O08786 P30551 P30552 P30553 P32238 P32239 P56481 P79266
Human
Rat
IC50: 124
Mouse
Ki: 22
Human
GENOME POLYPROTEIN A0A024B7W1 A0A0K1CY61 A0A0K2E2J2 A0A143MHK7 A0A1D8D5K2 A3EZI9 A3EZJ3 B0B3F0 C1KIQ2 D2K2A8 G1FEK8 I1U3K2 K7XGM7 K7XJL6 O39927 O39929 O92972 P03300 P03303 P03313 P06935 P12823 P12916 P14340 P17763 P19711 P26660 P26661 P26662 P26663 P26664 P27914 P27915 P27958 P29846 P29990 P29991 P33478 P69035 Q04045 Q0ZMF1 Q32ZE1 Q4U254 Q58HT7 Q66478 Q69422 Q6YMS4 Q7T664 Q80J95 Q81258 Q81495 Q82122 Q83883 Q91H74 Q91RS4 Q96662 Q99IB8 Q9WMX2 V5TFZ2
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Dengue virus 2
Dengue virus 1(Hawaii)
IC50: 10
Dengue virus 3 (strain S221/03)
IC50: 10
WNV
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
GERANYLGERANYL TRANSFERASE TYPE-1 SUBUNIT BETA P29702 P49354 P53609 P53610 Q04631 Q5EAD5 Q61239 Q8BUY9
Geranylgeranyl transferase type-1 subunit beta [A2V]/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha P49354 P53609
Human
Geranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha P29702 Q5EAD5
Bovine
IC50: 183
Geranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha P49354 P53609
Human
Human
Mouse
EC50: 6
Helicobacter pylori (strain J99 / ATCC 700824) (Campylobacter pylori J99)
IC50: 76
GLUTAMATE RECEPTOR A4FV91 B9V8S1 E1BGZ0 G1SXH9 O15399 Q00959 Q00960 Q00961 Q01097 Q12879 Q13224 Q14957 Q62645 Q62683
Human
Human
IC50: 33
GLUTAMATE RECEPTOR IONOTROPIC, NMDA 1 O15399 O60391 P35439 Q00959 Q00960 Q00961 Q01097 Q05586 Q12879 Q13224 Q14957 Q62645 Q8VHN2 Q9R1M7
Human
Human
Human
Human
Human
Human
Salmonella typhimurium (strain LT2 / SGSC1412 / ATCC 700720)
Ki: 1
Yeast
Escherichia coli (Enterobacteria)
GLUTATHIONE S-TRANSFERASE P O60341 O60674 O75116 O75460 P09211 P10415 P11362 P22607 P23458 P24864 P24941 P33981 P42330 P43405 Q13464 Q9BUB5 Q9UDY8
Human
Human
IC50: 81
Human
IC50: 41
Human
IC50: 25
Human
IC50: 132
Human
IC50: 96
Glutathione S-transferase P/Isoform 2 of Lysine-specific histone demethylase 1A (2) [158-876] O60341 P09211
Human
Glutathione S-transferase P/Isoform 2 of MAP kinase-interacting serine/threonine-protein kinase 1 (MNK1a) [T344D] P09211 Q9BUB5
Human
IC50: 110
Human
Human
IC50: 125
Glutathione S-transferase P/Mucosa-associated lymphoid tissue lymphoma translocation protein 1 P09211 Q9UDY8
Human
IC50: 48
Human
IC50: 11
Human
IC50: 10
Human
IC50: 182
GLYCOGEN SYNTHASE KINASE-3 BETA A0A059UE90 B2LUN4 G1T8E2 I6LNT8 I6YP72 P18266 P49840 P49841 P51136 Q9WV60
Human
Alpha-1,2-mannosidase/Alpha-1,2-mannosidase family protein/Alpha-1,2-mannosidase, putative/Glycoside hydrolase family 92/Putative alpha-1,2-mannosidase Q8A0C8 Q8A0C9 Q8A0E8 Q8A0M7 Q8A0N0 Q8A0N1 Q8A0Q6 Q8A0Q8 Q8A0Q9 Q8A113 Q8A182 Q8A193 Q8A1X8 Q8A1Y1 Q8A325 Q8A3K6 Q8A4H0 Q8A5N9 Q8A5X5 Q8A5Y1 Q8A6K3 Q8A6V7 Q8A8Y5
Bacteroides thetaiotaomicron
Ki: 1
Trypanosoma brucei brucei (strain 927/4 GUTat10.1)
IC50: 506
Neosartorya fumigata (Aspergillus fumigatus)
IC50: 27
Human
Human
IC50: 1
Human
Human
IC50: 244

