Target Names are taken from UniProtKB. To view the associated UniProt page, click on the UniProt ID. When we have data for a given Target in multiple species or for mutants of a given Target, we provide a header row (upper case, bold font) with all of the data followed by a separate for each species or variant of the Target.

Target Name  
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Target Name
Organism
Affinity Links
Articles
UniProts
Files
Rat
EC50: 8
Honeybee
IC50: 1
Human
Ki: 105 IC50: 497 Kd: 8 EC50: 602
Human
IC50: 568 Kd: 3 EC50: 342
Human
Ki: 5 IC50: 428 EC50: 78
Human
Ki: 72 IC50: 201 Kd: 1 EC50: 265
Fruit fly
IC50: 2 Kd: 6
HIV-1
IC50: 10
Avian erythroblastosis virus (strain ES4)
IC50: 15
Human immunodeficiency virus type 1
Kd: 2
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 6
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
IC50: 73
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 613 IC50: 915 Other: 20
Human immunodeficiency virus type 1
Ki: 131 IC50: 30
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 62
Human immunodeficiency virus type 1
Ki: 10 Other: 1
Human immunodeficiency virus type 1
Ki: 1
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 226 IC50: 43 EC50: 38
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus type 1
Ki: 8
Human immunodeficiency virus type 1
Ki: 367 IC50: 98
Human immunodeficiency virus type 1
Ki: 7
Human immunodeficiency virus 2
Ki: 16 IC50: 7
Human immunodeficiency virus type 1
IC50: 3
HIV-1
IC50: 1334 Kd: 8 EC50: 250
ALV-A RSA
EC50: 559
HIV-1
IC50: 28 Kd: 4 EC50: 79
HIV-1
Ki: 5 IC50: 84 EC50: 12
WMSV
Ki: 13 IC50: 22
RSV-Pr-C
IC50: 18 EC50: 8
Human immunodeficiency virus type 1
IC50: 132
Human immunodeficiency virus
Ki: 11 IC50: 52
Human immunodeficiency virus type 1
EC50: 83
Human immunodeficiency virus type 1
Ki: 2038 IC50: 2299 Kd: 84 EC50: 40 Koff: 39 Kon: 39
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus type 1
IC50: 84
Human immunodeficiency virus type 1
IC50: 32 EC50: 13
Human immunodeficiency virus type 1
Ki: 5 IC50: 5
Human immunodeficiency virus type 1
IC50: 42
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 5
Human immunodeficiency virus type 1
Ki: 3
Human immunodeficiency virus type 1
Ki: 5 IC50: 42 EC50: 12
Human immunodeficiency virus type 1
IC50: 1143
Human immunodeficiency virus type 1
Ki: 4 IC50: 57
Human immunodeficiency virus type 1
IC50: 181
Human immunodeficiency virus type 1
IC50: 9
Human immunodeficiency virus type 1
IC50: 10
Human immunodeficiency virus type 1
IC50: 10
Human immunodeficiency virus type 1
IC50: 296 Other: 5
Human immunodeficiency virus type 1
IC50: 9
Human immunodeficiency virus type 1
IC50: 155 Other: 1
Human immunodeficiency virus type 1
IC50: 56 Other: 3
Human immunodeficiency virus type 1
IC50: 18
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 1
Human immunodeficiency virus type 1
IC50: 43
Human immunodeficiency virus type 1
EC50: 6
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus type 1
ITC: 13
Human immunodeficiency virus type 1
Ki: 4 ITC: 4
Human immunodeficiency virus type 1
ITC: 5
Human immunodeficiency virus type 1
Ki: 4 ITC: 4
Human immunodeficiency virus type 1
Ki: 4 ITC: 4
Human immunodeficiency virus type 1
Ki: 4 ITC: 4
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus
EC50: 6
Human immunodeficiency virus type 1
ITC: 4
HIV-1
IC50: 2 EC50: 223
HTLV-1
Ki: 4 IC50: 27
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv)
IC50: 1
Human
IC50: 242
Mouse
IC50: 8
Human
Ki: 67 IC50: 25 Kd: 7
Human
Ki: 54 IC50: 134 Kd: 7 EC50: 22
Chicken
IC50: 18
Human
IC50: 746 Kd: 251
Rat
Kd: 4
Mus musculus
Kd: 4
Human
Kd: 22
Human
IC50: 1151 Kd: 730 EC50: 14
Mouse
IC50: 81 Kd: 19
Human
Kd: 71
Human
Kd: 85
Mouse
Kd: 4
Human
Kd: 210
Human
IC50: 17 Kd: 134
Human
IC50: 2
Human
Ki: 21 IC50: 21
Rat
Ki: 3
Human
Kd: 13
Enterococcus faecalis (strain ATCC 700802 / V583)
IC50: 44
HCV
Ki: 89 IC50: 140 EC50: 24
Hu/NV/NV/1968/US
EC50: 2
HCV
Ki: 300 IC50: 930 EC50: 305
HRV-1B
EC50: 7
DENV-1
IC50: 4 EC50: 15
Norovirus Hu/GII.P4_GII.4/Minerva
Ki: 19 IC50: 28
DENV-2
EC50: 9
HCV
IC50: 6 Other: 6
HCV
IC50: 19 EC50: 1
HCV
IC50: 1 EC50: 4
Hepacivirus C
IC50: 146
Hepatitis C Virus
Ki: 22 IC50: 100 Koff: 1 Kon: 1
Coxsackievirus B3 (strain Nancy)
Ki: 9 IC50: 103
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Ki: 241 IC50: 272 Kd: 41 EC50: 43
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Ki: 11
HCV
IC50: 225 EC50: 114
HCV
IC50: 189 EC50: 32
Hepacivirus C
Ki: 15 IC50: 197
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Ki: 10
HCV
IC50: 104 EC50: 428
HCV
Ki: 89 IC50: 400 EC50: 370
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Ki: 19 IC50: 8
Hepacivirus C
Ki: 63
ZIKV
IC50: 25 EC50: 9
ZIKV
IC50: 10 Kd: 4 EC50: 41
Human rhinovirus B
Ki: 167 IC50: 290 EC50: 144
Poliovirus type 1 (strain Mahoney)
IC50: 19 Kd: 1
Hepatitis GB virus B
IC50: 121
DENV-2
Ki: 115 IC50: 244 EC50: 137
WNV
Ki: 22 IC50: 284 Kd: 3
HRV-16
IC50: 9
Hepacivirus C
Ki: 36 IC50: 11
Dengue virus 2
Ki: 9 IC50: 61 Kd: 3
Norovirus Hu/GII.4-2002/WeertE022/2002/NL
IC50: 13
Norovirus Hu/GI/10360/2010/VNM
IC50: 13
Dengue virus
Ki: 5 IC50: 83 Kd: 2 EC50: 2
Hepacivirus C
Ki: 7 IC50: 7
Hepacivirus C
Ki: 2 Koff: 2 Kon: 2
HCV
Ki: 12 IC50: 67 EC50: 62
Dengue virus 3 (strain S221/03)
IC50: 10
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
IC50: 4 Kd: 4
HCV
IC50: 9 Kd: 10 EC50: 54 Koff: 10 Kon: 10
HCV
IC50: 7 Kd: 1 Koff: 1 Kon: 1
Hepatitis C virus genotype 1b (isolate Con1) (HCV)
Ki: 333 IC50: 219
Human
IC50: 53
Vibrio cholerae
IC50: 2
Human
Ki: 6
Human
Ki: 310 IC50: 1367 EC50: 174
Mouse
IC50: 101 EC50: 18
Rat
IC50: 97 Kd: 13 EC50: 9
Rhesus macaque
IC50: 1
Human
Ki: 116 IC50: 413 Kd: 89 EC50: 2557 Koff: 4
Crab-eating macaque
EC50: 4
Shiitake mushroom
IC50: 3
Aspergillus niger
Ki: 1 IC50: 1
Mucormycosis agent
Ki: 1 IC50: 1
Human
Ki: 1385 IC50: 4321 Kd: 13 EC50: 1516
Mouse
Ki: 1 IC50: 3 Kd: 4 EC50: 24
Rat
Ki: 28 IC50: 192 EC50: 112
Dog
Ki: 1 IC50: 4 EC50: 1
Trypanosoma cruzi (strain CL Brener)
Ki: 2 IC50: 35
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228)
IC50: 14
Streptococcus pneumoniae D39
IC50: 4
Lactobacillus fermentum
Ki: 4
Helicobacter pylori (strain J99 / ATCC 700824) (Campylobacter pylori J99)
IC50: 76
Enterococcus faecalis (strain ATCC 700802 / V583)
IC50: 33
Helicobacter pylori (strain ATCC 700392 / 26695) (Campylobacterpylori)
Ki: 1 IC50: 21 Kd: 3
African clawed frog
EC50: 3
Human
Ki: 142 IC50: 47 Kd: 4 EC50: 293
Rat
Ki: 101 IC50: 9 Kd: 1 EC50: 34
Rat
Ki: 169 IC50: 8 EC50: 31
Human
Ki: 57 IC50: 7 EC50: 28
Rat
Ki: 43 IC50: 7 EC50: 25
Human
Ki: 44 IC50: 4 EC50: 167
Pyrococcus horikoshii (strain ATCC 700860 / DSM 12428 / JCM 9974 /NBRC 100139 / OT-3)
Kd: 3
Onchocerca volvulus
Ki: 1
Escherichia coli (strain K12)
Ki: 4
Escherichia coli (strain K12)
Ki: 7 IC50: 7
Salmonella typhimurium (strain LT2 / SGSC1412 / ATCC 700720)
Ki: 1
Staphylococcus aureus
Ki: 11
Streptococcus pyogenes M1 GAS
IC50: 38
Human
Ki: 1
Escherichia coli (Enterobacteria)
Ki: 2 IC50: 2
Human
Ki: 4 IC50: 5
Baker's yeast
Ki: 1 IC50: 11
Plasmodium falciparum (isolate 3D7)
Ki: 1 IC50: 4
malaria parasite P. falciparum
IC50: 3
African malaria mosquito
IC50: 5
Schistosoma japonicum
IC50: 8
Crithidia fasciculata
Ki: 25 IC50: 22
malaria parasite P. falciparum
IC50: 42
Silk moth
Ki: 6 IC50: 6 Kd: 1 ITC: 4
Plasmodium falciparum (isolate 3D7)
IC50: 35
Social amoeba
IC50: 6
Human
Ki: 33 IC50: 251 EC50: 10
Human
Kd: 5
HHV-4
IC50: 835
Nipah virus
EC50: 7
malaria parasite P. vivax
IC50: 96
Trypanosoma brucei brucei (strain 927/4 GUTat10.1)
IC50: 506
Neosartorya fumigata (Aspergillus fumigatus)
IC50: 27
Plasmodium falciparum (isolate 3D7)
Ki: 32 IC50: 27
Baker's yeast
Ki: 12
Human
Ki: 23 IC50: 149
Human
Ki: 3
Human
Ki: 2 IC50: 328 Kd: 71 Koff: 2 Kon: 2 ITC: 10
Human
Ki: 1 IC50: 58 Kd: 4
Human
Ki: 34 IC50: 1741 Kd: 68 EC50: 13
Human
IC50: 3532 Kd: 302
Human
Ki: 1 IC50: 416
Salmonella newport
IC50: 3
Human
Ki: 12 IC50: 1
Yellow koji mold
IC50: 19

BDB Curated by BindingDB
EBI Curated by ChEMBL