PMID

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Article Title

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Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds.

University of Modena and Reggio Emilia

Synthesis, biological evaluation and molecular modeling of 1-oxa-4-thiaspiro- and 1,4-dithiaspiro[4.5]decane derivatives as potent and selective 5-HT

University of Modena and Reggio Emilia

Insights into the interaction of negative allosteric modulators with the metabotropic glutamate receptor 5: discovery and computational modeling of a new series of ligands with nanomolar affinity.

University of Modena and Reggio Emilia

Structure-affinity/activity relationships of 1,4-dioxa-spiro[4.5]decane based ligands ata<alpha>1 and 5-HT1A receptors.

University of Modena and Reggio Emilia

Exploring a potential palonosetron allosteric binding site in the 5-HT(3) receptor.

University of Modena and Reggio Emilia

2'-Deoxyuridine 5'-monophosphate substrate displacement in thymidylate synthase through 6-hydroxy-2H-naphtho[1,8-bc]furan-2-one derivatives.

University of Modena and Reggio Emilia

Ligand-based discovery of N-(1,3-dioxo-1H,3H-benzo[de]isochromen-5-yl)-carboxamide and sulfonamide derivatives as thymidylate synthase A inhibitors.

University of Modena and Reggio Emilia

Synthesis, biological evaluation, and docking studies of tetrahydrofuran- cyclopentanone- and cyclopentanol-based ligands acting at adrenergica1- and serotonine 5-HT1A receptors.

University of Modena and Reggio Emilia

Computational analysis of ligand recognition sites of homo- and heteropentameric 5-HT3 receptors.

University of Modena and Reggio Emilia

1,3-Dioxolane-based ligands incorporating a lactam or imide moiety: structure-affinity/activity relationship at alpha1-adrenoceptor subtypes and at 5-HT1A receptors.

University of Modena and Reggio Emilia

Discovery of a new series of 5-HT1A receptor agonists.

University of Modena and Reggio Emilia

Synthesis and structure-activity relationships of 1-aralkyl-4-benzylpiperidine and 1-aralkyl-4-benzylpiperazine derivatives as potent sigma ligands.

University of Modena and Reggio Emilia

Design, synthesis, biological evaluation and crystal structure determination of dual modulators of carbonic anhydrases and estrogen receptors.

University of Modena and Reggio Emilia

Dual Kinase-Bromodomain Inhibitors in Anticancer Drug Discovery: A Structural and Pharmacological Perspective.

University of Modena and Reggio Emilia

Folic Acid-Peptide Conjugates Combine Selective Cancer Cell Internalization with Thymidylate Synthase Dimer Interface Targeting.

University of Modena and Reggio Emilia

Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign.

University of Modena and Reggio Emilia

Novel Dithiolane-Based Ligands Combining Sigma and NMDA Receptor Interactions as Potential Neuroprotective Agents.

University of Modena and Reggio Emilia

SAR Studies and Biological Characterization of a Chromen-4-one Derivative as an Anti-

University of Modena and Reggio Emilia

Profiling of Flavonol Derivatives for the Development of Antitrypanosomatidic Drugs.

University of Modena and Reggio Emilia

Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic Infections.

University of Modena and Reggio Emilia

1,3-Dioxane as a scaffold for potent and selective 5-HT

University of Modena and Reggio Emilia

Isolation of a High-Affinity Cannabinoid for the Human CB1 Receptor from a Medicinal

University of Modena and Reggio Emilia

Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomics.

University of Modena and Reggio Emilia

1,2,4-Benzothiadiazine derivatives as alpha1 and 5-HT1A receptor ligands.

University of Modena and Reggio Emilia

Aryl thiosemicarbazones for the treatment of trypanosomatidic infections.

University of Modena and Reggio Emilia