Compile Data Set for Download or QSAR
Report error Found 87 Enz. Inhib. hit(s) with all data for entry = 50046319
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105834(CHEMBL3597594)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105833(CHEMBL3597593)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105801(CHEMBL3597596)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105802(CHEMBL3597597)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105801(CHEMBL3597596)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105833(CHEMBL3597593)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105805(CHEMBL3597600)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105805(CHEMBL3597600)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105803(CHEMBL3597598)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105802(CHEMBL3597597)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105833(CHEMBL3597593)
Affinity DataIC50: 0.400nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105832(CHEMBL3597592)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105837(CHEMBL3597585)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105803(CHEMBL3597598)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105806(CHEMBL3597602)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105834(CHEMBL3597594)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105831(CHEMBL3597584)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105831(CHEMBL3597584)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105832(CHEMBL3597592)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105834(CHEMBL3597594)
Affinity DataIC50: 0.800nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105831(CHEMBL3597584)
Affinity DataIC50: 0.900nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105844(CHEMBL3597586)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105805(CHEMBL3597600)
Affinity DataIC50: 1.30nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105837(CHEMBL3597585)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105802(CHEMBL3597597)
Affinity DataIC50: 1.80nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105832(CHEMBL3597592)
Affinity DataIC50: 2.80nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105806(CHEMBL3597602)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105803(CHEMBL3597598)
Affinity DataIC50: 3.80nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50149805(2-(Pyridin-3-yl)-5-(2-methylthiazol-4ylethynyl)pyr...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105832(CHEMBL3597592)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]R214127 from rat cloned mGluR1 receptor expressed in CHO-T-Rex cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50149805(2-(Pyridin-3-yl)-5-(2-methylthiazol-4ylethynyl)pyr...)
Affinity DataIC50: 6.10nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105806(CHEMBL3597602)
Affinity DataIC50: 9.70nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50084137(2-Methyl-6-phenylethynyl-pyridine | CHEMBL66654 | ...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105801(CHEMBL3597596)
Affinity DataIC50: 10nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50149805(2-(Pyridin-3-yl)-5-(2-methylthiazol-4ylethynyl)pyr...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50084137(2-Methyl-6-phenylethynyl-pyridine | CHEMBL66654 | ...)
Affinity DataIC50: 11nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50084137(2-Methyl-6-phenylethynyl-pyridine | CHEMBL66654 | ...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105803(CHEMBL3597598)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]R214127 from rat cloned mGluR1 receptor expressed in CHO-T-Rex cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105802(CHEMBL3597597)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]R214127 from rat cloned mGluR1 receptor expressed in CHO-T-Rex cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105839(CHEMBL3597595)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50122758(3-(2-(2-methylthiazol-4-yl)ethynyl)pyridine | 3-[(...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105838(FENOBAM)
Affinity DataIC50: 36nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMetabotropic glutamate receptor 1(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105832(CHEMBL3597592)
Affinity DataIC50: 39nMAssay Description:Negative allosteric modulatory activity at rat cloned mGluR1 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced calci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50122758(3-(2-(2-methylthiazol-4-yl)ethynyl)pyridine | 3-[(...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105833(CHEMBL3597593)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]R214127 from rat cloned mGluR1 receptor expressed in CHO-T-Rex cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105844(CHEMBL3597586)
Affinity DataIC50: 42nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105829(CHEMBL3597603)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50122758(3-(2-(2-methylthiazol-4-yl)ethynyl)pyridine | 3-[(...)
Affinity DataIC50: 47nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105844(CHEMBL3597586)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]R214127 from rat cloned mGluR1 receptor expressed in CHO-T-Rex cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 5(Human)
University of Modena and Reggio Emilia

Curated by ChEMBL
LigandPNGBDBM50105839(CHEMBL3597595)
Affinity DataIC50: 55nMAssay Description:Negative allosteric modulatory activity at human cloned mGluR5 receptor expressed in CHO-T-Rex cells assessed as inhibiton of quisqualate-induced cal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2016
Entry Details Article
PubMed
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