Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 12374
TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699087(4-(8-((2-fluoro-5-(trifluoromethyl)benzoyl)-D- val...)
Affinity DataIC50: 1.10nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699076(2-fluoro-N-((2R)-1-(4-(4-methoxyphenyl)-2- methyl-...)
Affinity DataIC50: 1.70nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699090(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-4-(p- tolyl)...)
Affinity DataIC50: 2.20nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699084(N-((2R)-1-(4-(4-fluorophenyl)-2-methyl-2,8- diazas...)
Affinity DataIC50: 3.40nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699100(2-fluoro-N-((2R)-3-methyl-1-oxo-1-(10-oxo-7- pheny...)
Affinity DataIC50: 3.5nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699072(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-1-oxo-4- phe...)
Affinity DataIC50: 3.80nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699056(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-1-oxo-4- phe...)
Affinity DataIC50: 4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699094(2-fluoro-N-((2R)-1-(4-(4-fluorophenyl)-2- methyl-2...)
Affinity DataIC50: 4.10nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699093(N-((1R)-1-cyclohexyl-2-(4-(4-fluorophenyl)-2- meth...)
Affinity DataIC50: 4.40nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699108(2-fluoro-N-((2R)-1-(7-(4-fluorophenyl)-9- methyl-3...)
Affinity DataIC50: 5.10nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699101(2-fluoro-N-((2R)-1-(7-(4-fluorophenyl)-10-oxo- 3,9...)
Affinity DataIC50: 6.5nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699061(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-4- phenyl-2,...)
Affinity DataIC50: 6.60nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699082(2-fluoro-N-((2R)-1-(4-(4-methoxyphenyl)-2- methyl-...)
Affinity DataIC50: 6.80nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699065(2-fluoro-N-((2R)-1-(4-(4-fluorophenyl)-2- methyl-1...)
Affinity DataIC50: 6.90nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699098(N-((2R)-1-(4-(4-fluorophenyl)-2-methyl-2,8- diazas...)
Affinity DataIC50: 6.90nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699063(N-((2R)-1-(4-(1H-indazol-5-yl)-2-methyl-2,8- diaza...)
Affinity DataIC50: 6.90nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699079(2-fluoro-N-((2R)-1-(4-(4-fluorophenyl)-2- methyl-2...)
Affinity DataIC50: 7.10nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699103(2-fluoro-N-((2R)-1-(7-(4-fluorophenyl)-9- methyl-1...)
Affinity DataIC50: 7.5nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699089(2-fluoro-N-((R)-1-((S)-4-(4-fluorophenyl)-2- methy...)
Affinity DataIC50: 7.80nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699083(2-fluoro-N-((2R)-1-(4-(4-methoxyphenyl)-2- methyl-...)
Affinity DataIC50: 9.30nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699107(2-fluoro-N-((2R)-3-methyl-1-(9-methyl-7- phenyl-3,...)
Affinity DataIC50: 9.90nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699071(2-fluoro-5-methyl-N-((2R)-3-methyl-1-(2- methyl-1-...)
Affinity DataIC50: 10.1nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699099(4-methyl-N-((2R)-3-methyl-1-(2-methyl-4- (pyridin-...)
Affinity DataIC50: 10.2nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699102(2-fluoro-N-((2R)-3-methyl-1-(9-methyl-10-oxo- 7-ph...)
Affinity DataIC50: 11.2nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699092(2-fluoro-N-((1R)-2-(4-(4-fluorophenyl)-2- methyl-2...)
Affinity DataIC50: 11.5nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699066(N-((2R)-1-(2-ethyl-4-(4-fluorophenyl)-1-oxo-2,8- d...)
Affinity DataIC50: 11.7nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699105(2-fluoro-N-((2S)-3-methyl-1-(9-methyl-10-oxo- 7-ph...)
Affinity DataIC50: 12nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699088(2-fluoro-N-((R)-1-((R)-4-(4-fluorophenyl)-2- methy...)
Affinity DataIC50: 12nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699058(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-1-oxo-4- (py...)
Affinity DataIC50: 13.3nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699062(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-4- (pyridin-...)
Affinity DataIC50: 13.4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699106(N-((2R)-3-methyl-1-(9-methyl-10-oxo-7-phenyl- 3,9-...)
Affinity DataIC50: 15.9nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699070(N-((2R)-3-methyl-1-(2-methyl-1-oxo-4-phenyl- 2,8-d...)
Affinity DataIC50: 16.4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699104(N-((2R)-1-(9-ethyl-7-(4-fluorophenyl)-10-oxo- 3,9-...)
Affinity DataIC50: 17.2nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699057(2-fluoro-N-((2R)-3-methyl-1-oxo-1-(1-oxo-4- phenyl...)
Affinity DataIC50: 19.2nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699064(2-fluoro-N-((2R)-1-(4-(4-fluorophenyl)-1-oxo- 2,8-...)
Affinity DataIC50: 22.6nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699067(2-fluoro-5-methoxy-N-((2R)-3-methyl-1-(2- methyl-1...)
Affinity DataIC50: 25.6nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699073(2-fluoro-N-((2R)-1-(4-(4-fluorophenyl)-2- isopropy...)
Affinity DataIC50: 34.2nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699091(N-((2R)-1-(4-(3,5-dimethylphenyl)-2-methyl-2,8- di...)
Affinity DataIC50: 40.4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699080(2-fluoro-N-((2R)-1-(4-(4-fluorophenyl)-2- isopropy...)
Affinity DataIC50: 44.4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699095(2,5-difluoro-N-((2R)-1-(4-(4-fluorophenyl)-2- meth...)
Affinity DataIC50: 47.3nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699097(N-((2R)-1-(4-(4-fluorophenyl)-2-methyl-2,8- diazas...)
Affinity DataIC50: 48.4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699068((R)-2-fluoro-N-(3-methyl-1-(2-methyl-1-oxo-4- phen...)
Affinity DataIC50: 55.6nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699059(2-fluoro-N-((2R)-3-methyl-1-oxo-1-(1-oxo-4- (pyrid...)
Affinity DataIC50: 56.2nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699060(N-((2R)-1-(4-(1H-indazol-5-yl)-2-methyl-1-oxo- 2,8...)
Affinity DataIC50: 58.9nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699085(methyl 8-((2-fluoro-5-(trifluoromethyl)benzoyl)- D...)
Affinity DataIC50: 59.7nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699069(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-1-oxo-4- phe...)
Affinity DataIC50: 66.8nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699055(N-((2R)-1-(2-(2-aminoethyl)-1,3-dioxo-4-phenyl- 2,...)
Affinity DataIC50: 69.8nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699074(N-((2R)-1-(2-(cyclopropylmethyl)-4-(4- fluoropheny...)
Affinity DataIC50: 73.4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699077(2-fluoro-N-((2R)-3-methyl-1-oxo-1-(2-oxo-4- phenyl...)
Affinity DataIC50: 74.4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetAutotaxin(Rat)
CADILA HEAL THCARE LIMITED

US Patent
LigandPNGBDBM699081(N-((2R)-1-(2-(cyclopropylmethyl)-4-(4- fluoropheny...)
Affinity DataIC50: 84.4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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