Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with Target = 'Sulfotransferase 2A1'
TargetSulfotransferase 2A1(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50380592(CHEMBL1552719)
Affinity DataIC50: 50nMAssay Description:Inhibition of ST (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSulfotransferase 2A1(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50427989(CHEMBL2325503)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of ST (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSulfotransferase 2A1(Rat)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM7462(cid_5280863 | CHEMBL150 | 3,5,7-trihydroxy-2-(4-hy...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSulfotransferase 2A1(Rat)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM23420(CHEMBL8145 | US8552057, 7 | 7-hydroxy-3-(4-hydroxy...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSulfotransferase 2A1(Rat)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSulfotransferase 2A1(Rat)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of rat SULT2A1-mediated dehydroepiandrosterone sulfonation incubated for 20 minsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSulfotransferase 2A1(Rat)
University of Bath

Curated by ChEMBL
LigandPNGBDBM50051828(2-(4-hydroxyphenyl)-3-methyl-1-(2,3,4,5,6-pentaflu...)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibitory activity against dehydroepiandrosterone sulfatase (DHA-STS)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSulfotransferase 2A1(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM50176062(3-(5H-dibenzo[a,d][7]annulen-5-yl)-N-methylpropan-...)
Affinity DataKi:  7.60E+4nM ΔG°:  -21.7kJ/molepH: 7.5 T: 2°CAssay Description:Reaction conditions were as follows: SULT1A1 or 2A1 (50 nM), PnP (3.0 or 100 uM, respectively; 2 x Km PnP), amoxipine or protriptyline (0, 50, 100, o...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSulfotransferase 2A1(Human)
Ocean University of China

Curated by ChEMBL
LigandPNGBDBM22870(CHEMBL1113 | Asendin | 2-chloro-11-piperazin-1-yld...)
Affinity DataKi:  1.25E+5nM ΔG°:  -20.6kJ/molepH: 7.5 T: 2°CAssay Description:Reaction conditions were as follows: SULT1A1 or 2A1 (50 nM), PnP (3.0 or 100 uM, respectively; 2 x Km PnP), amoxipine or protriptyline (0, 50, 100, o...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed