BDBM701110 (3aR,6aS)-5-(1-isopPropyl- 6-((4-phenyl-1H-imidazol-2- yl)ethynyl)-1H-pyrazolo[3,4- d]pyrimidin-4- yl)hexahydro-1H-furo[3,4- c]pyrrole::US20240343729, Example 25
SMILES CC(C)n1ncc2c(N3C[C@H]4COC[C@H]4C3)nc(C#Cc3nc(-c4ccccc4)c[nH]3)nc21
InChI Key InChIKey=JFCJLQOSZPVNTK-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 701110
TargetIsoform PDE10A2 of cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A (PDE10A2)(Human)
Benevolentai Cambridge
US Patent
Benevolentai Cambridge
US Patent
Affinity DataIC50: 0.112nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
Ligand InfoSimilars