BDBM701097 (3R)-3-Methyl-4-[2-[2-(1- methyl-4-phenyl-imidazol- 2-yl)ethynyl]-5,6,7,8- tetrahydropyrido[3,4- d]pyrimidin-4- yl]morpholine::US20240343729, Example 12
SMILES C[C@@H]1COCCN1c1nc(C#Cc2nc(-c3ccccc3)cn2C)nc2c1CCNC2
InChI Key InChIKey=JEMHMOJDFBAIRT-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 701097
TargetIsoform PDE10A2 of cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A (PDE10A2)(Human)
Benevolentai Cambridge
US Patent
Benevolentai Cambridge
US Patent
Affinity DataIC50: 0.0400nMAssay Description:Semi Log compound dilutions starting at a final concentration of 50 μM were dispensed into a black 384 well plate alongside, DMSO and an Inhibit...More data for this Ligand-Target Pair
Ligand InfoSimilars