BDBM576045 6-methyl-4-(2-methyl-1-(4- methylthio)benzyl)-1H-imidazo [4,5-b]pyridin-6-yl)-1H- pyrrolo[2,3-c]pyridin-7(6H)-one::US11466034, Example 3
SMILES CSc1ccc(Cn2c(C)nc3ncc(cc23)-c2cn(C)c(=O)c3[nH]ccc23)cc1
InChI Key InChIKey=GQDUGMPGNVUSLF-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 576045
Affinity DataIC50: 12.7nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:The assays of BRD4 (D1) and BRD4 (D2) were conducted in a 384-well polystyrene plate. The test compounds were first serially diluted in DMSO and the ...More data for this Ligand-Target Pair