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22 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
 
Diphenylborinic acid is a strong inhibitor of serine proteasesEBI
TBA
Small molecule inhibitors of PCSK9. SAR investigations of head and amine groups.EBI
Pfizer
Novel PCSK9 Inhibitors for Treating Cardiovascular Diseases.EBI
Smith, Gambrell & Russell
Structure-activity relationship and biological evaluation of xanthine derivatives as PCSK9 inhibitors for the treatment of atherosclerosis.EBI
Peking Union Medical College
Recent Update on the Development of PCSK9 Inhibitors for Hypercholesterolemia Treatment.EBI
Aligarh Muslim University
Inhibitors of Eukaryotic Translational Machinery as Therapeutic Agents.EBI
Merck
Potent Lys Patch-Containing Stapled Peptides Targeting PCSK9.EBI
University of Montpellier
Bioactive Cyclization Optimizes the Affinity of a Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9) Peptide Inhibitor.EBI
The University of Queensland
Discovery of Small-Molecule CD33 Pre-mRNA Splicing Modulators.EBI
Pfizer
A Series of Novel, Highly Potent, and Orally Bioavailable Next-Generation Tricyclic Peptide PCSK9 Inhibitors.EBI
Merck
From methylene bridged diindole to carbonyl linked benzimidazoleindole: Development of potent and metabolically stable PCSK9 modulators.EBI
University of Wisconsin-Madison
Series of Novel and Highly Potent Cyclic Peptide PCSK9 Inhibitors Derived from an mRNA Display Screen and Optimized via Structure-Based Design.EBI
Merck
Novel Cyclic Tetramer Compounds as PCSK9 Inhibitors for Treating Metabolic Disorders.EBI
Lauren Mccallister
Discovery of 2,3'-diindolylmethanes as a novel class of PCSK9 modulators.EBI
University of Wisconsin
Small molecules as inhibitors of PCSK9: Current status and future challenges.EBI
China Pharmaceutical University
Small molecule modulators of PCSK9 - A literature and patent overview.EBI
Astrazeneca
O'-(epoxyalkyl)tyrosines and (epoxyalkyl)phenylalanine as irreversible inactivators of serine proteases: synthesis and inhibition mechanism.EBI
State University
Highly active CSF1R inhibitor compoundBDB
Xiamen Biotime Biotechnology
Isoquinoline amine compounds as mGluR4 allosteric potentiators, compositions, and methods of treating neurological dysfunctionBDB
Vanderbilt University
Toll-like receptor 7 (TLR7) agonists having heteroatom-linked aromatic moieties, conjugates thereof, and methods and uses thereforBDB
Bristol-Myers Squibb
Glucagon receptor modulatorsBDB
Pfizer
Biosynthesis and recycling of nicotinamide cofactors in mycobacterium tuberculosis. An essential role for NAD in nonreplicating bacilli.BDB
National Institutes of Health