Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50015060
TargetProprotein convertase subtilisin/kexin type 9(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50582341(CHEMBL5092750)
Affinity DataKd:  974nMAssay Description:Binding affinity to full length C-terminal Avi/His6-tagged human PCSK9 expressed in Expi293 cells assessed as equilibrium dissociation constant by su...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 9(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50582342(CHEMBL5088175)
Affinity DataKd:  660nMAssay Description:Binding affinity to human PCSK9 assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 9(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50582341(CHEMBL5092750)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of tEGF-A[HA] binding to biotinylated human PCSK9 incubated for 2 hrs by ELISA based competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed