29 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Article Title
Organization
Bishomoisoprenoid triazole bisphosphonates as inhibitors of geranylgeranyl diphosphate synthase.
University of Iowa
Phosphinophosphonates and Their Tris-pivaloyloxymethyl Prodrugs Reveal a Negatively Cooperative Butyrophilin Activation Mechanism.
University of Iowa
Potent Triazole Bisphosphonate Inhibitor of Geranylgeranyl Diphosphate Synthase.
University of Iowa
N-Oxide derivatives of 3-(3-pyridyl)-2-phosphonopropanoic acids as potential inhibitors of Rab geranylgeranylation.
University of Iowa
Geranyl and neryl triazole bisphosphonates as inhibitors of geranylgeranyl diphosphate synthase.
University of Iowa
Mono- and dialkyl isoprenoid bisphosphonates as geranylgeranyl diphosphate synthase inhibitors.
University of Iowa
Pivaloyloxymethyl-modified isoprenoid bisphosphonates display enhanced inhibition of cellular geranylgeranylation.
University of Iowa
Structure-activity studies on a potent antagonist to organophosphate-induced toxicity.
University of Iowa
Opioid receptor probes derived from cycloaddition of the hallucinogen natural product salvinorin A.
University of Iowa
Synthesis and biological evaluation of a series of aromatic bisphosphonates.
University of Iowa
Rapid computational identification of the targets of protein kinase inhibitors.
University of Iowa
Impact of α-modifications on the activity of triazole bisphosphonates as geranylgeranyl diphosphate synthase inhibitors.
University of Iowa
Amides as bioisosteres of triazole-based geranylgeranyl diphosphate synthase inhibitors.
University of Iowa
Deacylcortivazol-like pyrazole regioisomers reveal a more accommodating expanded binding pocket for the glucocorticoid receptor.
University of Iowa
Synthesis and Metabolism of BTN3A1 Ligands: Studies on Modifications of the Allylic Alcohol.
University of Iowa
Identification of an ethyl 5,6-dihydropyrazolo[1,5-c]quinazoline-1-carboxylate as a catalytic inhibitor of DNA gyrase.
University of Iowa
Inhibition of HIV integrase by novel nucleotides bearing tricyclic bases.
University of Iowa
Probing structural requirements for human topoisomerase I inhibition by a novel N1-Biphenyl fluoroquinolone.
University of Iowa
Novel benzimidazole phosphonates as potential inhibitors of protein prenylation.
University of Iowa
Synthesis and Bioactivity of the Alanyl Phosphonamidate Stereoisomers Derived from a Butyrophilin Ligand.
University of Iowa
Phosphonamidate Prodrugs of a Butyrophilin Ligand Display Plasma Stability and Potent Vγ9 Vδ2 T Cell Stimulation.
University of Iowa
Natural Products Discovered in a High-Throughput Screen Identified as Inhibitors of RGS17 and as Cytostatic and Cytotoxic Agents for Lung and Prostate Cancer Cell Lines.
University of Iowa
α-Methylation enhances the potency of isoprenoid triazole bisphosphonates as geranylgeranyl diphosphate synthase inhibitors.
University of Iowa
Design, synthesis, and evaluation of novel N-1 fluoroquinolone derivatives: Probing for binding contact with the active site tyrosine of gyrase.
University of Iowa
