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26 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Conformationally Defined Rexinoids and Their Efficacy in the Prevention of Mammary Cancers.EBI
University of Alabama At Birmingham
Potent inhibition of human sulfotransferase 1A1 by 17a-ethinylestradiol: role of 3'-phosphoadenosine 5'-phosphosulfate binding and structural rearrangements in regulating inhibition and activity.EBI
University of Alabama At Birmingham
Methyl substitution of a rexinoid agonist improves potency and reveals site of lipid toxicity.EBI
University of Alabama At Birmingham
Methyl-substituted conformationally constrained rexinoid agonists for the retinoid X receptors demonstrate improved efficacy for cancer therapy and prevention.EBI
University of Alabama At Birmingham
Pyrrolidinobenzoic acid inhibitors of influenza virus neuraminidase: the hydrophobic side chain influences type A subtype selectivity.EBI
University of Alabama At Birmingham
Identification of novel inhibitors of bacterial surface enzyme Staphylococcus aureus Sortase A.EBI
University of Alabama At Birmingham
Tethered dimers as NAD synthetase inhibitors with antibacterial activity.EBI
University of Alabama At Birmingham
3-Amino-5,5-dimethylhexanoic acid. Synthesis, resolution, and effects on carnitine acyltransferases.EBI
University of Alabama At Birmingham
Virtual screening to identify lead inhibitors for bacterial NAD synthetase (NADs).EBI
University of Alabama At Birmingham
Synthesis and Structure-Activity Relationships of 5'-Aryl-14-alkoxypyridomorphinans: Identification of a μ Opioid Receptor Agonist/δ Opioid Receptor Antagonist Ligand with Systemic Antinociceptive Activity and Diminished Opioid Side Effects.EBI
University of Alabama At Birmingham
Potent inhibition of influenza sialidase by a benzoic acid containing a 2-pyrrolidinone substituent.EBI
University of Alabama At Birmingham
Conformationally defined retinoic acid analogues. 4. Potential new agents for acute promyelocytic and juvenile myelomonocytic leukemias.EBI
University of Alabama At Birmingham
Conformationally defined 6-s-trans-retinoic acid analogs. 3. Structure-activity relationships for nuclear receptor binding, transcriptional activity, and cancer chemopreventive activity.EBI
University of Alabama At Birmingham
A conformationally defined 6-s-trans-retinoic acid isomer: synthesis, chemopreventive activity, and toxicity.EBI
University of Alabama At Birmingham
Conformationally defined 6-s-trans-retinoic acid analogs. 2. Selective agonists for nuclear receptor binding and transcriptional activity.EBI
University of Alabama At Birmingham
Comparative molecular field analysis of hydantoin binding to the neuronal voltage-dependent sodium channel.EBI
University of Alabama At Birmingham
Effects of log P and phenyl ring conformation on the binding of 5-phenylhydantoins to the voltage-dependent sodium channel.EBI
University of Alabama At Birmingham
Bicyclic hydantoins with a bridgehead nitrogen. Comparison of anticonvulsant activities with binding to the neuronal voltage-dependent sodium channel.EBI
University of Alabama At Birmingham
Discovery and evaluation of nNaEBI
University of Alabama At Birmingham
(Hetero)aryl cyclopropylamine compounds as LSD1 inhibitorsBDB
Oryzon Genomics
Substituted spiropiperidinyl compounds useful as GPR120 agonistsBDB
Merck Sharp & Dohme
Process for making isoquinoline compoundsBDB
Fibrogen
Methyl-pyrrolidine ether derivativesBDB
Hoffmann-La Roche
1,2,6-substituted benzimidazoles as flap modulatorsBDB
Janssen Pharmaceutica
Fluoro-olefins as peptidomimetic inhibitors of dipeptidyl peptidases.BDB
University of Antwerp