Compile Data Set for Download or QSAR
Report error Found 98 Enz. Inhib. hit(s) with all data for entry = 1591
TargetDipeptidyl peptidase 4(Human)
University of Antwerp

LigandPNGBDBM12466(1-[(1-Adamantylamino)acetyl]-2-pyrrolidinecarbonit...)
Affinity DataIC50: 350nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12437(9.8k | 1-Benzyl-N-(2-cyclohexylidene-2-fluoroethyl...)
Affinity DataIC50: 1.04E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12425(9.7g | 1-Benzyl-N-(2-cyclopentylidene-2-fluoroethy...)
Affinity DataIC50: 1.30E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp

LigandPNGBDBM12465(1-{[(2-Phenylethyl)amino]acetyl}-2-pyrrolidinecarb...)
Affinity DataIC50: 2.13E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12455(1-Benzyl-N-[2-oxo-2-(1-piperidinyl)ethyl]-4-piperi...)
Affinity DataIC50: 3.10E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp

LigandPNGBDBM12467(17c | 1-{[(4-Fluorobenzyl)amino]acetyl}-2-pyrrolid...)
Affinity DataIC50: 3.70E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12436(N-(2-Cyclohexylidene-2-fluoroethyl)- 4-piperidinam...)
Affinity DataIC50: 4.20E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12442((2H-1,3-benzodioxol-5-ylmethyl)(2-cyclopentylidene...)
Affinity DataIC50: 7.50E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12434(N-(2-Cyclohexylidene-2-fluoroethyl)-N-[3-(trifluor...)
Affinity DataIC50: 9.60E+3nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12422((2-cyclopentylidene-2-fluoroethyl)[(4-fluorophenyl...)
Affinity DataIC50: 1.08E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12435(N-(2-Cyclohexylidene-2-fluoroethyl)-N-(2-phenyleth...)
Affinity DataIC50: 1.10E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp

LigandPNGBDBM12460(11.7b/1 | (2Z)-2-[2-(adamantan-1-ylamino)-1-fluoro...)
Affinity DataIC50: 1.20E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12438(9.8l | benzyl 4-[(2-cyclohexylidene-2-fluoroethyl)...)
Affinity DataIC50: 1.28E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12432(9.8f | N-(1,3-Benzodioxol-5-ylmethyl)-2-cyclohexyl...)
Affinity DataIC50: 1.29E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12431(N-(2-Cyclohexylidene-2-fluoroethyl)-N-(4-methoxybe...)
Affinity DataIC50: 1.34E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12451(10.8c | (2H-1,3-benzodioxol-5-ylmethyl)(2-cyclohex...)
Affinity DataIC50: 1.44E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp

LigandPNGBDBM12463((1R,S)-(2E)-2-[2-(1-Adamantylamino)-1-fluoroethyli...)
Affinity DataIC50: 1.50E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12421(N-(2-Cyclopentylidene-2-fluoroethyl)-N-(4-methoxyb...)
Affinity DataIC50: 1.55E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12423(N-(2-Cyclopentylidene-2-fluoroethyl)-N-(2-pyridiny...)
Affinity DataIC50: 1.57E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12465(1-{[(2-Phenylethyl)amino]acetyl}-2-pyrrolidinecarb...)
Affinity DataIC50: 1.63E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12433((2-cyclohexylidene-2-fluoroethyl)[(4-fluorophenyl)...)
Affinity DataIC50: 2.19E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12467(17c | 1-{[(4-Fluorobenzyl)amino]acetyl}-2-pyrrolid...)
Affinity DataIC50: 2.55E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12441(benzyl(2-cyclopentylideneethyl)amine | 10.7b | Ole...)
Affinity DataIC50: 2.60E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12424(9.7f | N-(2-Cyclopentylidene-2-fluoroethyl)-N-(2-p...)
Affinity DataIC50: 2.72E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12459((1R,S)-(2Z)-2-{1-Fluoro-2-[(2-phenylethyl)amino]et...)
Affinity DataIC50: 3.29E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12430(benzyl(2-cyclohexylidene-2-fluoroethyl)amine | 9.8...)
Affinity DataIC50: 3.40E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12462((1R,S)-(2E)-2-{1-Fluoro-2-[(2-phenylethyl)amino]et...)
Affinity DataIC50: 3.61E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12420(N-Benzyl-2-cyclopentylidene-2-fluoroethanamine | 9...)
Affinity DataIC50: 3.78E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12464((1R,S)-(2E)-2-{1-Fluoro-2-[(4-fluorobenzyl)amino]e...)
Affinity DataIC50: 4.04E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12458(N-(1,3-benzodioxol-5-ylmethyl)-N-(2-piperidin-1-yl...)
Affinity DataIC50: 4.20E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12457(N-Benzyl-2-thioxo-2-(1-piperidinyl)ethaneamine | b...)
Affinity DataIC50: 4.84E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12454(15.2c | 2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1...)
Affinity DataIC50: 5.20E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12426(9.7h | (2-cyclopentylidene-2-fluoroethyl)[3-(dimet...)
Affinity DataIC50: 5.37E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12439(9.8m | N-(2-Cyclohexylidene-2-fluoroethyl)-N3,N3-d...)
Affinity DataIC50: 5.46E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12450(10.8b | benzyl(2-cyclohexylideneethyl)amine | Olef...)
Affinity DataIC50: 5.53E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12440(N-(2-cyclopentylideneethyl)cyclohexanamine | 10.7a...)
Affinity DataIC50: 6.20E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12445(15.1c | 2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1...)
Affinity DataIC50: 6.30E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12448(N-(1,3-benzodioxol-5-ylmethyl)-N-(2-pyrrolidin-1-y...)
Affinity DataIC50: 6.70E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12456(N-[2-(piperidin-1-yl)-2-sulfanylideneethyl]cyclohe...)
Affinity DataIC50: 6.90E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12461((2Z)-2-(1-fluoro-2-{[(4-fluorophenyl)methyl]amino}...)
Affinity DataIC50: 8.73E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12419(N-(2-cyclopentylidene-2-fluoroethyl)cyclohexanamin...)
Affinity DataIC50: 9.00E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12428(N-(2-cyclohexylidene-2-fluoroethyl)adamantan-1-ami...)
Affinity DataIC50: 9.13E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12446(16.1a | N-Cyclohexyl-2-thioxo-2-(1-pyrrolidinyl)et...)
Affinity DataIC50: 9.20E+4nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12429(N-(2-Cyclohexylidene-2-fluoroethyl)aniline | 9.8c ...)
Affinity DataIC50: 1.00E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12460(11.7b/1 | (2Z)-2-[2-(adamantan-1-ylamino)-1-fluoro...)
Affinity DataIC50: 1.00E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12463((1R,S)-(2E)-2-[2-(1-Adamantylamino)-1-fluoroethyli...)
Affinity DataIC50: 1.00E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp

LigandPNGBDBM12434(N-(2-Cyclohexylidene-2-fluoroethyl)-N-[3-(trifluor...)
Affinity DataIC50: 1.25E+5nMpH: 8.3 T: 2°CAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 4(Human)
University of Antwerp

LigandPNGBDBM12438(9.8l | benzyl 4-[(2-cyclohexylidene-2-fluoroethyl)...)
Affinity DataIC50: 1.25E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12466(1-[(1-Adamantylamino)acetyl]-2-pyrrolidinecarbonit...)
Affinity DataIC50: 1.34E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDipeptidyl peptidase 2(Human)
University of Antwerp

LigandPNGBDBM12449(N-(2-cyclohexylideneethyl)cyclohexanamine | 10.8a ...)
Affinity DataIC50: 1.36E+5nMAssay Description:The DPP inhibition was measured by monitoring the cleavage of chromogenic substrate in the presence of each inhibitor compound. IC50 value was determ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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