28 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Chemoenzymatic synthesis and binding affinity of novel (R)- and (S)-3-aminomethyl-1-tetralones, potential atypical antipsychotics.
Universidad De Santiago De Compostela
Potent and selective MAO-B inhibitory activity: amino- versus nitro-3-arylcoumarin derivatives.
Universidad De Santiago De Compostela
Synthesis and biological evaluation of a series of aminoalkyl-tetralones and tetralols as dual dopamine/serotonin ligands.
Universidad De Santiago De Compostela
Synthesis and binding affinity of new 1,4-disubstituted triazoles as potential dopamine D(3) receptor ligands.
Universidad De Santiago De Compostela
Synthesis and binding affinity of potential atypical antipsychotics with the tetrahydroquinazolinone motif.
Universidad De Santiago De Compostela
Synthesis, binding affinity, and molecular docking analysis of new benzofuranone derivatives as potential antipsychotics.
Universidad De Santiago De Compostela
Butyrophenone analogues in the carbazole series: synthesis and determination of affinities at D2 and 5-HT2A receptors.
Universidad De Santiago De Compostela
Synthesis and biological evaluation of 1a,25-dihydroxyvitamin D3 analogues with a long side chain at C12 and short C17 side chains.
Universidad De Santiago De Compostela
On a possible neutral charge state for the catalytic dyad inß-secretase when bound to hydroxyethylene transition state analogue inhibitors.
Universidad De Santiago De Compostela
A prodrug approach for improving antituberculosis activity of potent Mycobacterium tuberculosis type II dehydroquinase inhibitors.
Universidad De Santiago De Compostela
MAO inhibitory activity modulation: 3-Phenylcoumarins versus 3-benzoylcoumarins.
Universidad De Santiago De Compostela
New halogenated phenylcoumarins as tyrosinase inhibitors.
Universidad De Santiago De Compostela
New halogenated 3-phenylcoumarins as potent and selective MAO-B inhibitors.
Universidad De Santiago De Compostela
Synthesis and biological evaluation of new nanomolar competitive inhibitors of Helicobacter pylori type II dehydroquinase. Structural details of the role of the aromatic moieties with essential residues.
Universidad De Santiago De Compostela
Synthesis and evaluation of 6-methyl-3-phenylcoumarins as potent and selective MAO-B inhibitors.
Universidad De Santiago De Compostela
Synthesis, binding affinity and SAR of new benzolactam derivatives as dopamine D3 receptor ligands.
Universidad De Santiago De Compostela
6-N,N-dimethylamino-2,3-naphthalimide: a new environment-sensitive fluorescent probe in delta- and mu-selective opioid peptides.
Universidad De Santiago De Compostela
Pyridazines part 41: synthesis, antiplatelet activity and SAR of 2,4,6-substituted 5-(3-oxo-3-phenylprop-1-en-1-yl)- or 5-(3-phenylprop-2-enoyl)pyridazin-3(2H)-ones.
Universidad De Santiago De Compostela
Design, synthesis, and vasorelaxant and platelet antiaggregatory activities of coumarin-resveratrol hybrids.
Universidad De Santiago De Compostela
Ligand recognition by RAR and RXR receptors: binding and selectivity.
Universidad De Santiago De Compostela
Structure-based design, synthesis, and biological evaluation of inhibitors of Mycobacterium tuberculosis type II dehydroquinase.
Universidad De Santiago De Compostela
Parallel solid-phase synthesis and evaluation of inhibitors of Streptomyces coelicolor type II dehydroquinase.
Universidad De Santiago De Compostela
Exploring the water-binding pocket of the type II dehydroquinase enzyme in the structure-based design of inhibitors.
Universidad De Santiago De Compostela
Experimental and 'in silico' analysis of the effect of pH on HIV-1 protease inhibitor affinity: implications for the charge state of the protein ionogenic groups.
Universidad De Santiago De Compostela
Synthesis and binding affinity of new pyrazole and isoxazole derivatives as potential atypical antipsychotics.
Universidad De Santiago De Compostela
25 S-Adamantyl-23-yne-26,27-dinor-1α,25-dihydroxyvitamin D
Universidad De Santiago De Compostela
