Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50007643
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50018958(CHEBI:75401 | QUINPIROLE)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human D2S receptor expressed in CHOK1 cells assessed as inhibition of forskolin induced cAMP production preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50018958(CHEBI:75401 | QUINPIROLE)
Affinity DataEC50:  151nMAssay Description:Agonist activity at human D2S receptor expressed in CHOK1 cells assessed as inhibition of forskolin induced cAMP production preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50511120(CHEMBL4591554)
Affinity DataEC50:  2.95E+3nMAssay Description:Agonist activity at human D2S receptor expressed in CHOK1 cells assessed as inhibition of forskolin induced cAMP production preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50492966(CHEMBL2414991)
Affinity DataEC50:  1.02E+4nMAssay Description:Agonist activity at human D2S receptor expressed in CHOK1 cells assessed as inhibition of forskolin induced cAMP production preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50511120(CHEMBL4591554)
Affinity DataEC50:  2.95E+3nMAssay Description:Agonist activity at human D2S receptor expressed in CHOK1 cells assessed as inhibition of forskolin induced cAMP production preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50492966(CHEMBL2414991)
Affinity DataEC50:  1.02E+4nMAssay Description:Agonist activity at human D2S receptor expressed in CHOK1 cells assessed as inhibition of forskolin induced cAMP production preincubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  5.16nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50511120(CHEMBL4591554)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50511120(CHEMBL4591554)
Affinity DataKi:  197nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50511120(CHEMBL4591554)
Affinity DataKi:  286nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50511120(CHEMBL4591554)
Affinity DataKi:  288nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50492966(CHEMBL2414991)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50492966(CHEMBL2414991)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50492966(CHEMBL2414991)
Affinity DataKi:  832nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50492966(CHEMBL2414991)
Affinity DataKi:  838nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO-K1 cells by radioligand competitive binding analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed