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25 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Structural optimization, biological evaluation, and application of peptidomimetic prostate specific antigen inhibitors.EBI
The Johns Hopkins University
Potent, selective and low-calcemic inhibitors of CYP24 hydroxylase: 24-sulfoximine analogues of the hormone 1alpha,25-dihydroxyvitamin D(3).EBI
The Johns Hopkins University
Synthesis and biochemical evaluation of triazole/tetrazole-containing sulfonamides against thrombin and related serine proteases.EBI
The Johns Hopkins University
Low-calcemic, highly antiproliferative, 23-oxa ether analogs of the natural hormone 1 alpha,25-dihydroxyvitamin D3: design, synthesis, and preliminary biological evaluation.EBI
The Johns Hopkins University
Design, Synthesis, and Evaluation of 4- and 5-Substituted EBI
The Johns Hopkins University
Ferrochelatase inhibitors and methods of useBDB
Indiana University
N-SUBSTITUTED INDOLE DERIVATIVES AS SEROTONERGIC AGENTS USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETOBDB
Mindset Pharma
IRE1 small molecule inhibitorsBDB
Cornell University
INHIBITOR OF ENHANCER OF ZESTE HOMOLOGUE 2, AND USE THEREOFBDB
Haisco Pharmaceuticals
Pyrazolyl pyrimidinylamine compounds as CDK2 inhibitorsBDB
Incyte
Bcl-2 inhibitorsBDB
Beigene
Therapeutic heterocyclic compoundsBDB
Gilead Sciences
6-(5-membered heteroaryl)isoquinolin-3-yl-(5-membered heteroaryl) carboxamides and preparation and use thereofBDB
Samumed
Inhibitors of plasma kallikrein and uses thereofBDB
Shire Human Genetic Therapies
Pyrrolo[2,3-d]pyrimidinyl, pyrrolo[2,3-b]pyrazinyl and pyrrolo[2,3-d]pyridinyl acrylamidesBDB
Pfizer
Pyrimidine compounds as inhibitors of protein kinases IKK epsilon and/or TBK-1, processes for their preparation, and pharmaceutical compositions containing themBDB
Domainex
Coupling of metabotropic glutamate receptors 2 and 4 to G alpha 15, G alpha 16, and chimeric G alpha q/i proteins: characterization of new antagonists.BDB
Upr Centre
Benzimidazole inhibitors of the sodium channelBDB
Degiacomo, Interim Trustee, Mark G.
N-4-Pyrimidinyl-1H-indazol-4-amine inhibitors of Lck: indazoles as phenol isosteres with improved pharmacokinetics.BDB
Gsk
Heteroaryl compounds and uses thereofBDB
Celgene Car
Synthesis of indoleamine 2,3-dioxygenase inhibitory analogues of the sponge alkaloid exiguamine a.BDB
University of British Columbia
Ethynyl derivativesBDB
Hoffmann-La Roche
Benzamide derivativeBDB
Chugai Seiyaku Kabushiki Kaisha