Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 2559
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21978(1H-indol-4-ol | 4-hydroxyindole, 18)
Affinity DatapH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21983(3-(2-aminoethyl)-5,10-diphenyl-1H,4H,11H-anthracen...)
Affinity DatapH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21975((4S)-16'-(2-aminoethyl)-9'-hydroxy-1,3,6',6'-tetra...)
Affinity DataKi:  41nM ΔG°:  -43.9kJ/molepH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21979(4,7-dihydro-1H-indole-4,7-dione | Indolequinone, 1...)
Affinity DataKi:  190nM ΔG°:  -39.9kJ/molepH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21982(3-(2-aminoethyl)-5-(3-methyl-2,5-dioxo-1-propylimi...)
Affinity DataKi:  200nM ΔG°:  -39.8kJ/molepH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21981(methyl 4-[3-(2-{[(benzyloxy)carbonyl]amino}ethyl)-...)
Affinity DataKi:  260nM ΔG°:  -39.1kJ/molepH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21984(methyl 4-{4,7-dioxo-3-[2-(3-phenylpropanamido)ethy...)
Affinity DataKi:  260nM ΔG°:  -39.1kJ/molepH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21980(methyl 4-(4,7-dioxo-4,7-dihydro-1H-indol-5-yl)-3-m...)
Affinity DataKi:  420nM ΔG°:  -37.9kJ/molepH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21976(benzyl N-[2-(4,7-dioxo-4,7-dihydro-1H-indol-3-yl)e...)
Affinity DataKi:  1.49E+3nM ΔG°:  -34.6kJ/molepH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21977(benzyl N-{2-[5-(1,3-dioxo-2-phenyl-2,3-dihydro-1H-...)
Affinity DataKi:  1.09E+4nM ΔG°:  -29.5kJ/molepH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIndoleamine 2,3-dioxygenase 1(Human)
University of British Columbia

LigandPNGBDBM21973(2-amino-3-(1-methyl-1H-indol-3-yl)propanoic acid |...)
Affinity DataKi:  6.20E+4nM ΔG°:  -25.0kJ/molepH: 6.5 T: 2°CAssay Description:The ability of the compounds prepared in this study to inhibit purified recombinant human IDO was evaluated with a steady state spectrophotometric as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed