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31 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Identification of the First Selective Activin Receptor-Like Kinase 1 Inhibitor, a Reversible Version of L-783277.EBI
Korea University
Synthesis and in vitro antiproliferative activity of C5-benzyl substituted 2-amino-pyrrolo[2,3-d]pyrimidines as potent Hsp90 inhibitors.EBI
Korea University
Design, synthesis and biological evaluation of PSMA/hepsin-targeted heterobivalent ligands.EBI
Korea University
Syringaresinol induces mitochondrial biogenesis through activation of PPARß pathway in skeletal muscle cells.EBI
Korea University
Structure-based design, synthesis, and biological evaluation of Leu-Arg dipeptide analogs as novel hepsin inhibitors.EBI
Korea University
Synthesis and biological evaluation of 3-phenethylazetidine derivatives as triple reuptake inhibitors.EBI
Korea University
trans-Caryophyllene is a natural agonistic ligand for peroxisome proliferator-activated receptor-a.EBI
Korea University
Exploration of 3-Aminoazetidines as Triple Reuptake Inhibitors by Bioisosteric Modification of 3-a-Oxyazetidine.EBI
Korea University
The dipeptide H-Trp-Glu-OH (WE) shows agonistic activity to peroxisome proliferator-activated protein-a and reduces hepatic lipid accumulation in lipid-loaded H4IIE cells.EBI
Korea University
Cyanidin, a natural flavonoid, is an agonistic ligand for liver X receptor alpha and beta and reduces cellular lipid accumulation in macrophages and hepatocytes.EBI
Korea University
Induction of ABCA1 and ABCG1 expression by the liver X receptor modulator cineole in macrophages.EBI
Korea University
Ethyl 2,4,6-trihydroxybenzoate is an agonistic ligand for liver X receptor that induces cholesterol efflux from macrophages without affecting lipid accumulation in HepG2 cells.EBI
Korea University
Discovery of potent and selective rhodanine type IKKß inhibitors by hit-to-lead strategy.EBI
Korea University
Polyhydroxylated macrolides from Seimatosporium discosioides and their effects on the activation of peroxisome proliferator-activated receptor gamma.EBI
Korea University
Acetylenic acid analogues from the edible mushroom Chanterelle (Cantharellus cibarius) and their effects on the gene expression of peroxisome proliferator-activated receptor-gamma target genes.EBI
Korea University
Ursolic acid is a PPAR-a agonist that regulates hepatic lipid metabolism.EBI
Korea University
Synthesis and 11ß hydroxysteroid dehydrogenase 1 inhibition of thiazolidine derivatives with an adamantyl group.EBI
Korea University
Discovery of cyclicsulfonamide derivatives as 11beta-hydroxysteroid dehydrogenase 1 inhibitors.EBI
Korea University
Discovery of a NADPH oxidase inhibitor, (E)-3-cyclohexyl-5-(4-((2-hydroxyethyl)(methyl)amino)benzylidene)-1-methyl-2-thioxoimidazolidin-4-oneone, as a novel therapeutic for Parkinson's disease.EBI
Korea University
Identification of Pyridinyltriazine Derivatives as Potent panFGFR Inhibitors against Gatekeeper Mutants for Overcoming Drug Resistance.EBI
Korea University
Novel Macrocyclic Peptidomimetics Targeting the Polo-Box Domain of Polo-Like Kinase 1.EBI
Korea University
Anti-glioma effects of 2-aminothiophene-3-carboxamide derivatives, ANO1 channel blockers.EBI
Korea University
Discovery and Characterization of Pure RhlR Antagonists against EBI
Korea University
Anti-inflammatory Metabolites from EBI
Korea University
Identification of Novel Resorcinol Amide Derivatives as Potent and Specific Pyruvate Dehydrogenase Kinase (PDHK) Inhibitors.EBI
Korea University
Benzylideneacetone Derivatives Inhibit Osteoclastogenesis and Activate Osteoblastogenesis Independently Based on Specific Structure-Activity Relationship.EBI
Korea University
Novel β- and γ-Amino Acid-Derived Inhibitors of Prostate-Specific Membrane Antigen.EBI
Korea University
Identification of a Unique Resorcylic Acid Lactone Derivative That Targets Both Lymphangiogenesis and Angiogenesis.EBI
Korea University
Design, synthesis, and biological evaluation of novel aminopyrimidinylisoindolines as AXL kinase inhibitors.EBI
Korea University
Spiroindole Alkaloids and Spiroditerpenoids from Aspergillus duricaulis and Their Potential Neuroprotective Effects.EBI
Korea University
First SAR Study for Overriding NRAS Mutant Driven Acute Myeloid Leukemia.EBI
Korea University