Compile Data Set for Download or QSAR
Report error Found 121 Enz. Inhib. hit(s) with all data for entry = 50016724
TargetFibroblast growth factor receptor 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50355393(CHEMBL1834657 | US9434697, BGJ398 | US9730931, BGJ...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR1 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596830(CHEMBL5179166)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR1 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596831(CHEMBL5177100)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR1 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596832(CHEMBL5198569)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR1 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596833(CHEMBL5193966)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR1 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596834(CHEMBL5181852)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR1 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50355393(CHEMBL1834657 | US9434697, BGJ398 | US9730931, BGJ...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR2 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596830(CHEMBL5179166)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR2 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR2 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM301310(3-(2,6-difluoro-3,5-dimethoxyphenyl)-1-ethyl-8-(mo...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR2 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596831(CHEMBL5177100)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR2 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596832(CHEMBL5198569)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR2 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596833(CHEMBL5193966)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR2 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596834(CHEMBL5181852)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR2 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596833(CHEMBL5193966)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596833(CHEMBL5193966)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596852(CHEMBL5193739)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50355393(CHEMBL1834657 | US9434697, BGJ398 | US9730931, BGJ...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FGFR3 K650E mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596830(CHEMBL5179166)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FGFR3 K650E mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596831(CHEMBL5177100)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FGFR3 K650E mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596832(CHEMBL5198569)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FGFR3 K650E mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596833(CHEMBL5193966)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FGFR3 K650E mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596834(CHEMBL5181852)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of FGFR3 K650E mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596831(CHEMBL5177100)
Affinity DataIC50: 0.520nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596832(CHEMBL5198569)
Affinity DataIC50: 0.580nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596831(CHEMBL5177100)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596832(CHEMBL5198569)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50355393(CHEMBL1834657 | US9434697, BGJ398 | US9730931, BGJ...)
Affinity DataIC50: 0.660nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50355393(CHEMBL1834657 | US9434697, BGJ398 | US9730931, BGJ...)
Affinity DataIC50: 0.680nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596830(CHEMBL5179166)
Affinity DataIC50: 0.920nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM301310(3-(2,6-difluoro-3,5-dimethoxyphenyl)-1-ethyl-8-(mo...)
Affinity DataIC50: 0.970nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596834(CHEMBL5181852)
Affinity DataIC50: 0.980nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596850(CHEMBL5200941)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596851(CHEMBL5204120)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of wild-type FGFR1 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596829(CHEMBL5194218)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of wild-type FGFR2 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM301310(3-(2,6-difluoro-3,5-dimethoxyphenyl)-1-ethyl-8-(mo...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of wild-type FGFR1 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596830(CHEMBL5179166)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596852(CHEMBL5193739)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596849(CHEMBL5174975)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596837(CHEMBL5203040)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596834(CHEMBL5181852)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50525939(Balversa | Erdafitinib | Jnj-42756493)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of FGFR3 K650E mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 3(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596829(CHEMBL5194218)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of wild-type FGFR3 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596842(CHEMBL5206623)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM301310(3-(2,6-difluoro-3,5-dimethoxyphenyl)-1-ethyl-8-(mo...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 1(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596829(CHEMBL5194218)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of wild-type FGFR1 (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596850(CHEMBL5200941)
Affinity DataIC50: 4nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetFibroblast growth factor receptor 2(Human)
Korea University

Curated by ChEMBL
LigandPNGBDBM50596843(CHEMBL5185122)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of FGFR2 N549H mutant (unknown origin) by radiometric kinase activity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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