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22 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Allosteric Glutaminase Inhibitors Based on a 1,4-Di(5-amino-1,3,4-thiadiazol-2-yl)butane Scaffold.EBI
Johns Hopkins University
D-Amino acid oxidase inhibitors based on the 5-hydroxy-1,2,4-triazin-6(1H)-one scaffold.EBI
Johns Hopkins University
6-Hydroxy-1,2,4-triazine-3,5(2H,4H)-dione Derivatives as Novel D-Amino Acid Oxidase Inhibitors.EBI
Johns Hopkins University
Structure-Metabolism Relationships in the Glucuronidation of d-Amino Acid Oxidase Inhibitors.EBI
Johns Hopkins University
d-Thiolactones as prodrugs of thiol-based glutamate carboxypeptidase II (GCPII) inhibitors.EBI
Johns Hopkins University
Synthesis of kojic acid derivatives as secondary binding site probes of D-amino acid oxidase.EBI
Johns Hopkins University
Design, synthesis, and pharmacological evaluation of bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide 3 (BPTES) analogs as glutaminase inhibitors.EBI
Johns Hopkins University
Pharmacophore modeling strategies for the development of novel nonsteroidal inhibitors of human aromatase (CYP19).EBI
Johns Hopkins University
Inhibition of xc¿?¿ transporter-mediated cystine uptake by sulfasalazine analogs.EBI
Johns Hopkins University
Applying linear interaction energy method for rational design of noncompetitive allosteric inhibitors of the sarco- and endoplasmic reticulum calcium-ATPase.EBI
Johns Hopkins University
Discovery and Evaluation of Novel Angular Fused Pyridoquinazolinonecarboxamides as RNA Polymerase I Inhibitors.EBI
Johns Hopkins University
Allosteric kidney-type glutaminase (GLS) inhibitors with a mercaptoethyl linker.EBI
Johns Hopkins University
Neutral sphingomyelinase 2 inhibitors based on the 4-(1H-imidazol-2-yl)-2,6-dialkoxyphenol scaffold.EBI
Johns Hopkins University
Peptidomimetics of Arg-Phe-NH2 as small molecule agonists of Mas-related gene C (MrgC) receptors.EBI
Johns Hopkins University
Recent advances in the development of polyamine analogues as antitumor agents.EBI
Johns Hopkins University
Application of a flexible synthesis of (5R)-thiolactomycin to develop new inhibitors of type I fatty acid synthase.EBI
Johns Hopkins University
Amino pyrimidine SSAO inhibitorsBDB
Eli Lilly
Pyrimidines and use thereofBDB
Purdue Pharma
Pyrrolo[2,3-d]pyrimidine compounds as inhibitors of protein kinasesBDB
Acea Biosciences
Substituted tricyclic compounds and methods of use thereofBDB
Bayer Intellectual Property
Benzimidazole inhibitors of the sodium channelBDB
SRMLSC