The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 3.0M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 695K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

If BindingDB was of value to your research, please take a moment to donate to this nonprofit project. Your donation will let us provide you with more data and improved service.

Advanced Search

18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Functional characterization of the human multidrug transporter, ABCG2, expressed in insect cells.EBI
Hungarian Academy of Sciences
Design, synthesis, pharmacological evaluation, and structure-activity study of novel endomorphin analogues with multiple structural modifications.EBI
Hungarian Academy of Sciences
Synthesis of heteroaromatic tropeines and heterogeneous binding to glycine receptors.EBI
Hungarian Academy of Sciences
Validation of high-affinity binding sites for succinic acid through distinguishable binding of gamma-hydroxybutyric acid receptor-specific NCS 382 antipodes.EBI
Hungarian Academy of Sciences
New endomorphin analogues containing alicyclic beta-amino acids: influence on bioactive conformation and pharmacological profile.EBI
Hungarian Academy of Sciences
Beta-methyl substitution of cyclohexylalanine in Dmt-Tic-Cha-Phe peptides results in highly potent delta opioid antagonists.EBI
Hungarian Academy of Sciences
Discovery of selective fragment-sized immunoproteasome inhibitors.EBI
Hungarian Academy of Sciences
The impact of binding site waters on the activity/selectivity trade-off of Janus kinase 2 (JAK2) inhibitors.EBI
Hungarian Academy of Sciences
Deltorphin II analogues with 6-hydroxy-2-aminotetralin-2-carboxylic acid in position 1.EBI
Hungarian Academy of Sciences
Conformationally constrained deltorphin analogs with 2-aminotetralin-2-carboxylic acid in position 3.EBI
Hungarian Academy of Sciences
Synthesis of tropeines and allosteric modulation of ionotropic glycine receptors.EBI
Hungarian Academy of Sciences
Inhibition of the LOX enzyme family members with old and new ligands. Selectivity analysis revisited.EBI
Hungarian Academy of Sciences
Discovery of d-amino acid oxidase inhibitors based on virtual screening against the lid-open enzyme conformation.EBI
Hungarian Academy of Sciences
Discovery of isatin and 1H-indazol-3-ol derivatives as d-amino acid oxidase (DAAO) inhibitors.EBI
Hungarian Academy of Sciences
Spiro[pyrrolidine-3,3'-oxindoles] as 5-HTEBI
Hungarian Academy of Sciences
Indole derivatives and their use in neurodegenerative diseasesBDB
Merck Patent
Substituted pyrazolo[3,4-d]pyrimidines as kinase inhibitorsBDB
Principia Biopharma