Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50019193
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202498(H-Dmt-Tic-(2S,3S)-beta-MeCha-Phe-OH | CHEMBL219482)
Affinity DataKi:  0.480nMAssay Description:Displacement of [3H]Ile5,6-deltorphin from delta opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202505(H-Tyr-Tic-Cha-Phe-OH | CHEMBL197937)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]Ile5,6-deltorphin from delta opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202506(H-Dmt-Tic-(2R,3S)-beta-MeCha-Phe-OH | CHEMBL376453)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]Ile5,6-deltorphin from delta opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202500(H-Dmt-Tic-(2R,3R)-beta-MeCha-Phe-OH | CHEMBL375094)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]Ile5,6-deltorphin from delta opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202502(H-Dmt-Tic-(2S,3R)-beta-MeCha-Phe-OH | CHEMBL375095)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]Ile5,6-deltorphin from delta opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202507(H-Dmt-Tic-(2S,3S)-beta-MeCha-Phe-NH2 | CHEMBL26931...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]Ile5,6-deltorphin from delta opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202501(H-Dmt-Tic-(2S,3R)-beta-MeCha-Phe-NH2 | CHEMBL41542...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]Ile5,6-deltorphin from delta opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202504(H-Dmt-Tic-(2R,3S)-beta-MeCha-Phe-NH2 | CHEMBL21878...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]Ile5,6-deltorphin from delta opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202503(H-Dmt-Tic-(2R,3R)-beta-MeCha-Phe-NH2 | CHEMBL21878...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]Ile5,6-deltorphin from delta opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202506(H-Dmt-Tic-(2R,3S)-beta-MeCha-Phe-OH | CHEMBL376453)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202501(H-Dmt-Tic-(2S,3R)-beta-MeCha-Phe-NH2 | CHEMBL41542...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202504(H-Dmt-Tic-(2R,3S)-beta-MeCha-Phe-NH2 | CHEMBL21878...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202502(H-Dmt-Tic-(2S,3R)-beta-MeCha-Phe-OH | CHEMBL375095)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202503(H-Dmt-Tic-(2R,3R)-beta-MeCha-Phe-NH2 | CHEMBL21878...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202507(H-Dmt-Tic-(2S,3S)-beta-MeCha-Phe-NH2 | CHEMBL26931...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202500(H-Dmt-Tic-(2R,3R)-beta-MeCha-Phe-OH | CHEMBL375094)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202498(H-Dmt-Tic-(2S,3S)-beta-MeCha-Phe-OH | CHEMBL219482)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50202505(H-Tyr-Tic-Cha-Phe-OH | CHEMBL197937)
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed