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TargetHistone deacetylase 1/3/4/6/7(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047416(CHEMBL3319215)
Affinity DataIC50: 3.60nMAssay Description:Displacement of [125I]human ghrelin from rat GHS-R1a expressed in HEK cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50588304(CHEMBL5202398)
Affinity DataIC50: 5nMAssay Description:Inhibition of rat HDAC1 using Boc-Lys(Ac)-AMC as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50154337(6-((9S,13aR)-5-(S)-1-Benzyl-8,8-dimethyl-4,7,10,13...)
Affinity DataIC50: 21nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375534(CHEMBL259517)
Affinity DataIC50: 130nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50082665(4-(dimethylamino)-N-(7-(hydroxyamino)-7-oxoheptyl)...)
Affinity DataIC50: 240nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50115659((S)-3-biphenyl-4-yl-2-(7-hydroxycarbamoyl-heptanoy...)
Affinity DataIC50: 440nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375542(CHEMBL261492)
Affinity DataIC50: 570nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375540(CHEMBL259708)
Affinity DataIC50: 590nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375548(CHEMBL259434)
Affinity DataIC50: 630nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375543(CHEMBL261272)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375545(CHEMBL260080)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375537(CHEMBL261587)
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375541(CHEMBL409860)
Affinity DataIC50: 2.55E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375539(CHEMBL264926)
Affinity DataIC50: 3.01E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375535(CHEMBL264411)
Affinity DataIC50: 3.03E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375536(CHEMBL409526)
Affinity DataIC50: 3.18E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375546(CHEMBL406734)
Affinity DataIC50: 3.19E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375544(CHEMBL263884)
Affinity DataIC50: 5.19E+3nMAssay Description:Inhibition of HDAC1 in rat liver extract by trypsin assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375538(CHEMBL427776)
Affinity DataIC50: 7.53E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Rat)
Chengdu University of Traditional Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50375547(CHEMBL259826)
Affinity DataIC50: 8.76E+3nMAssay Description:Inhibition of HDAC1 in rat liver extractMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed