Compile Data Set for Download or QSAR
Report error Found 787 for UniProtKB: Q13936
LigandPNGBDBM50016385(CHEMBL158853 | 4-Methyl-2-(3-nitro-phenyl)-2,5-dih...)
Affinity DataKd:  360nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels of guinea pig myocardiumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50015432(CHEMBL39925 | 6-Methyl-2-methylsulfanyl-4-(3-nitro...)
Affinity DataKd:  23nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50318494(3-ethyl 5-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,...)
Affinity DataKd:  0.260nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50035793(6-Methyl-2-methylsulfanyl-4-(2-methylsulfanyl-phen...)
Affinity DataKd:  1.52E+3nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035794(4-Methyl-2-methylsulfanyl-13-nitro-3,8,9,10,11,16b...)
Affinity DataKd:  5nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035796(2-Methylsulfanyl-4-(3-nitro-phenyl)-4,7-dihydro-1H...)
Affinity DataKd:  3.69E+4nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035798(4-(2-Butylsulfanyl-phenyl)-2-methylsulfanyl-4,7-di...)
Affinity DataKd: >5.00E+4nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035797(4-Methyl-2-methylsulfanyl-15-nitro-3,8,9,10,11,16b...)
Affinity DataKd:  873nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035801(2-Methylsulfanyl-4-(2-methylsulfanyl-5-nitro-pheny...)
Affinity DataKd: >5.00E+4nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035799(2-Methylsulfanyl-4-(2-methylsulfanyl-3-nitro-pheny...)
Affinity DataKd:  1.37E+4nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035790(6-Methyl-2-methylsulfanyl-4-(2-methylsulfanyl-3-ni...)
Affinity DataKd:  30nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035802(6-Methyl-2-methylsulfanyl-4-(2-methylsulfanyl-5-ni...)
Affinity DataKd:  2.70E+3nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035800(CHEMBL283013 | CHEMBL105672 | (S)-2,6-Dimethyl-5-n...)
Affinity DataKd:  18nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035791(2-Methylsulfanyl-4-(2-methylsulfanyl-phenyl)-4,7-d...)
Affinity DataKd:  4.52E+4nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035789(6-Methyl-2-methylsulfanyl-4-(3-nitro-phenyl)-1,4-d...)
Affinity DataKd:  480nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50035795(4-Methyl-2-methylsulfanyl-3,8,9,10,11,16b-hexahydr...)
Affinity DataKd:  18nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataKd:  0.400nMAssay Description:Displacement of [3H]nitrendipine from dihydropyridine receptor of guinea pig myocardial membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50226808(CHEMBL3392278)
Affinity DataKd:  3.40E+3nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50226760(CHEMBL2398396)
Affinity DataKd:  12nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50227245(CHEMBL3392281)
Affinity DataKd:  2.60nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50226978(CHEMBL282279)
Affinity DataKd:  120nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50226804(CHEMBL88149)
Affinity DataKd:  105nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50226761(CHEMBL3392285)
Affinity DataKd:  35nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel in guinea pig ventricular myocardium membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50016388(CHEMBL345843 | 5-(2-Dimethylamino-ethyl)-4-methyl-...)
Affinity DataKd:  488nMAssay Description:Inhibition of [3H]nitrendipine binding to calcium channels of guinea pig myocardiumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50538344(CHEMBL4633246)
Affinity DataEC50: >3.30E+4nMAssay Description:Inhibition of human Cav1.2 by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
LigandPNGBDBM720548(US20250051345, Example 1)
Affinity DataEC50:  220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720549(US20250051345, Example 2)
Affinity DataEC50:  61nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720550(US20250051345, Example 3)
Affinity DataEC50:  2.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720551(US20250051345, Example 4)
Affinity DataEC50:  2.90E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720552(US20250051345, Example 5)
Affinity DataEC50: >2.60E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720553(US20250051345, Example 6)
Affinity DataEC50:  250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720554(BayK8644 | US20250051345, Comparative Example 1)
Affinity DataEC50:  21nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720555(RS30124 | US20250051345, Comparative Example 2)
Affinity DataEC50:  450nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720556(CGP028392 | US20250051345, Comparative Example 3)
Affinity DataEC50:  280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720557(CAS 85825-32-7 | US20250051345, Comparative Exampl...)
Affinity DataEC50:  2.24E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720558(CAS 85825-31-6 | US20250051345, Comparative Exampl...)
Affinity DataEC50:  360nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720559(CAS 92638-18-1 | US20250051345, Comparative Exampl...)
Affinity DataEC50:  510nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM720560(US20250051345, Comparative Example 7)
Affinity DataEC50:  930nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
Go to US Patent

LigandPNGBDBM50227255(CHEMBL102907)
Affinity DataIC50: 0.00810nMAssay Description:Inhibition of [3H]nitrendipine binding to guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details Article
PubMed
LigandPNGBDBM50227481(CHEMBL286157)
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel of guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50227261(CHEMBL317044)
Affinity DataIC50: 0.0130nMAssay Description:Inhibition of [3H]nitrendipine binding to guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details Article
PubMed
LigandPNGBDBM50227259(CHEMBL441428)
Affinity DataIC50: 0.0150nMAssay Description:Inhibition of [3H]nitrendipine binding to guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details Article
PubMed
LigandPNGBDBM50227474(CHEMBL286598)
Affinity DataIC50: 0.0170nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel of guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50227478(CHEMBL37402)
Affinity DataIC50: 0.0220nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel of guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50227256(CHEMBL103806)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of [3H]nitrendipine binding to guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2018
Entry Details Article
PubMed
LigandPNGBDBM50227480(CHEMBL37899)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel of guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50227476(CHEMBL204616)
Affinity DataIC50: 0.0330nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel of guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50227479(CHEMBL35368)
Affinity DataIC50: 0.0450nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel of guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50227473(CHEMBL1099207)
Affinity DataIC50: 0.0460nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel of guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
LigandPNGBDBM50227475(CHEMBL285868)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of [3H]nitrendipine binding to L-type calcium channel of guinea pig ileal longitudinal smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
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