TargetGuanine nucleotide-binding protein G(q) subunit alpha(Human)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Inhibition of Galphaq/11 (unknown origin)More data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(q) subunit alpha/subunit alpha-11(Human)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of G-alphaq/11 in human platelet rich plasma assessed as inhibition of ADP-mediated platelet aggregationMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(q) subunit alpha(Human)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of G-alphaq/11 in human platelet rich plasma assessed as inhibition of ADP-mediated calcium ion mobilizationMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(q) subunit alpha(Human)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of Galphaq/11 (unknown origin)More data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(q) subunit alpha(Human)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of wild type GNAQ (unknown origin) expressed in CRISPR/Cas9 engineered HEK293 cellsMore data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(q) subunit alpha(Human)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 2.26E+4nMAssay Description:Inhibition of Galphaq/11 (unknown origin) expressed in CHO cells coexpressing M1 receptor assessed as reduction in carbachol-induced IP1 accumulation...More data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(q) subunit alpha(Human)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 4.86E+4nMAssay Description:Inhibition of Galphaq/11 (unknown origin) expressed in CHO cells coexpressing M1 receptor assessed as reduction in carbachol-induced IP1 accumulation...More data for this Ligand-Target Pair
TargetGuanine nucleotide-binding protein G(q) subunit alpha(Human)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 5.52E+4nMAssay Description:Binding affinity to Galphaq/11 (unknown origin) expressed in HEK293 cells cotransfected with AT1R/Galphaq-RLuc8/ Ggamma2-venus/Gbeta1 assessed as inh...More data for this Ligand-Target Pair
