Compile Data Set for Download or QSAR
Report error Found 5 of affinity data for UniProtKB/TrEMBL: P50135
TargetHistamine N-methyltransferase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM586429(Amodiaquin | USRE49340, Rank 6 | BDBM50041457)
Affinity DataKi:  19nMAssay Description:Inhibition of histamine N-methyltransferase by radiochemical assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetHistamine N-methyltransferase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50026331(L-2-Amino-4-[5-(6-amino-purin-9-yl)-3,4-dihydroxy-...)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition constant was evaluated against Histamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine N-methyltransferase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50026331(L-2-Amino-4-[5-(6-amino-purin-9-yl)-3,4-dihydroxy-...)
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition constant was evaluated against Histamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine N-methyltransferase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataKi:  1.81E+4nMAssay Description:Inhibition constant was evaluated against Histamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine N-methyltransferase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataKi:  1.81E+4nMAssay Description:Inhibition constant was evaluated against Histamine N-methyl-transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed