Affinity DataKd: 100nMAssay Description:Binding affinity towards Vasopressin V2 receptor in LLCPK cellsMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity towards Vasopressin V2 receptor in LLCPK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 uM in LLCPKI cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMAssay Description:Tested for the inhibition to V2 subtype receptor using [3H]- (VS2) as radioligand at 3 nM and arginine-vasopressin at 2 uM in LLCPKI cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Ability to displace [3H]AVP from Vasopressin V2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Compound was tested for its ability to inhibit binding of arginine vasopressin to Vasopressin receptor (V1 subtype)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Compound was tested for its ability to inhibit binding of arginine vasopressin to Vasopressin receptor (V1 subtype)More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of LVP stimulated adenylate cyclase activity in pig kidney medullary membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of LVP stimulated adenylate cyclase activity in pig kidney medullary membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of LVP stimulated adenylate cyclase activity in pig kidney medullary membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:In vitro antagonist activity was measured by inhibition of vasopressin-stimulated adenylate cyclase in renal medullary preparation in humanMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Compound was tested for inhibition against V2 vasopressin receptor in pig renal medullary membrane preparations.More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of LVP stimulated adenylate cyclase activity in pig kidney medullary membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Compound was tested for inhibition against V2 vasopressin receptor in pig renal medullary membrane preparations.More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Inhibition of LVP stimulated adenylate cyclase activity in pig kidney medullary membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Compound was tested for inhibition against V2 vasopressin receptor in pig renal medullary membrane preparations.More data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Inhibition of LVP stimulated adenylate cyclase activity in pig kidney medullary membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Compound was tested for inhibition against V2 vasopressin receptor in pig renal medullary membrane preparations.More data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Tested for inhibition of vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of LVP-sensitive adenylate cyclase in a pig renal medullary preparationMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of LVP stimulated adenylate cyclase activity in pig kidney medullary membraneMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of LVP stimulated adenylate cyclase activity in pig kidney medullary membraneMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition constant for vasopressin-stimulated adenylate cyclase of medullary membranes of pig kidney (Vasopressin V2 receptor)More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Tested for inhibition of [3H]LVP binding to vasopressin receptor in medullary membranes of pig kidney.More data for this Ligand-Target Pair
