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Report error Found 30 of affinity data for UniProtKB/TrEMBL: P32241
LigandPNGBDBM50435130(CHEMBL1893324)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at VPAC1 in human SH-SY5Y cells assessed as cAMP accumulation incubated for 60 mins by Eu-cAMP tracer based LANCE ultra cAMP assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50606527(CHEMBL5220770)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at VPAC1 in human SH-SY5Y cells assessed as cAMP accumulation incubated for 60 mins by Eu-cAMP tracer based LANCE ultra cAMP assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50200209(CHEMBL219499)
Affinity DataEC50:  0.600nMAssay Description:Activity at human VPAC1 receptor in CHO cells by measuring cAMP accumulationMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50250019(PACAP | PACAP-38 | CHEMBL524658 | PACAP(1-38) | PA...)
Affinity DataIC50: 0.0400nMAssay Description:Displacement of [125I]PACAP1-27 from human recombinant PAC1 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50250019(PACAP | PACAP-38 | CHEMBL524658 | PACAP(1-38) | PA...)
Affinity DataIC50: 0.0500nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50435130(CHEMBL1893324)
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]VIP from human recombinant VIP1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50208990(CHEMBL3884667)
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]VIP from human recombinant VPAC1 receptor expressed in CHO cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50435130(CHEMBL1893324)
Affinity DataIC50: 0.120nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50435130(CHEMBL1893324)
Affinity DataIC50: 0.120nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM392076(US10301272, Example 7/9)
Affinity DataIC50: 0.470nMAssay Description:Displacement of [125I]VIP from human recombinant VPAC1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50250018(PACAP27 | CHEMBL524852)
Affinity DataIC50: 5.90nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50498951(CHEMBL3736134)
Affinity DataIC50: 9nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50498951(CHEMBL3736134)
Affinity DataIC50: 9.30nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50498950(CHEMBL3736230)
Affinity DataIC50: 11nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50498950(CHEMBL3736230)
Affinity DataIC50: 12nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50200209(CHEMBL219499)
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]PACAP27 from human VPAC1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50250074([Bip6]PACAP27 | CHEMBL507480)
Affinity DataIC50: 14nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50606528(CHEMBL5219662)
Affinity DataIC50: 118nMAssay Description:Antagonist activity at VPAC1 in human SH-SY5Y cells assessed as inhibition of PACAP38-induced cAMP accumulation pre-incubated for 30 mins followed by...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50360601(CHEMBL1933349 | MK-0893)
Affinity DataIC50: 1.16E+4nMAssay Description:Antagonist activity at human VPAC1 expressed in HT-29 cells assessed as inhibition of glucagon-induced cAMP accumulation preincubated for 30 mins pri...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50435130(CHEMBL1893324)
Affinity DataKi:  0.0670nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM81828(CAS_37221-79-7 | VIP(4-28) | Vasoactive intestinal...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM81828(CAS_37221-79-7 | VIP(4-28) | Vasoactive intestinal...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM86051(NSC_0 | CAS_0 | [Lys15, Arg16, Leu27]VIP(1-7)GRF(8...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM81828(CAS_37221-79-7 | VIP(4-28) | Vasoactive intestinal...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM86051(NSC_0 | CAS_0 | [Lys15, Arg16, Leu27]VIP(1-7)GRF(8...)
Affinity DataKi:  7.70nMMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM86051(NSC_0 | CAS_0 | [Lys15, Arg16, Leu27]VIP(1-7)GRF(8...)
Affinity DataKi:  8.90nMMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM86050(Ac-L-His-L-Ser-L-Asp-L-Ala-L-Val-L-Phe-L-Thr-L-Glu...)
Affinity DataKi:  1.02E+3nMMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM86050(Ac-L-His-L-Ser-L-Asp-L-Ala-L-Val-L-Phe-L-Thr-L-Glu...)
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM86694(N'-(3-Chloro-4-morpholinophenyl)-N-hydroxyform...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50122872(4-Amino-5-chloro-2,3-dihydro-benzofuran-7-carboxyl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed