Compile Data Set for Download or QSAR
Report error Found 119 of affinity data for UniProtKB/TrEMBL: P30082
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataEC50:  8nMAssay Description:cAMP accumulation in rat hepatocytes in the presence rolipramMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059356([des-His1, Nle6, Glu9] glucagon-NH2 | CHEMBL236999...)
Affinity DataKd:  501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059365([des-Phe6, Glu9] glucagon-NH2 | CHEMBL412352)
Affinity DataKd:  631nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059354([des-Phe6] glucagon-NH2 | CHEMBL438574)
Affinity DataKd:  501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059360([des-His1, des-Phe6] glucagon-NH2 | CHEMBL429198)
Affinity DataKd:  562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059351([des-His1, des-Phe6, Glu9] glucagon | [des-Phe6, G...)
Affinity DataKd:  794nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059355([des-Phe6] glucagon | CHEMBL409611)
Affinity DataKd:  562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059361([des-His1, des-Phe6] glucagon | CHEMBL439271)
Affinity DataKd:  708nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059357([des-His1, Asp6, Glu9] glucagon-NH2 | CHEMBL438218)
Affinity DataKd:  501nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50087844(c[ Lys12, Asp21] glucagon-NH2 | CHEMBL266411)
Affinity DataEC50:  794nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataEC50:  5nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50087848(c[Asp15, Lys18,] glucagon-NH2 | CHEMBL427644)
Affinity DataEC50:  320nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059362([des-His1, des-Phe6, Glu9] glucagon-NH2 | CHEMBL26...)
Affinity DataKd:  6.31nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059358([des-His1, Tyr6,Glu9] glucagon-NH2 | CHEMBL267885)
Affinity DataKd:  631nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059359([des-His1, des-Gly4, Glu9] glucagon-NH2 | CHEMBL41...)
Affinity DataKd:  891nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059363([des-His1,Ala6, Glu9] glucagon-NH2 | CHEMBL437095)
Affinity DataKd:  398nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059352([des-His1, Trp6, Glu9] glucagon-NH2 | CHEMBL442499)
Affinity DataKd:  562nMAssay Description:pA2 value against Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50557260(CHEMBL4741000)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at rat glucagon receptor expressed in HEK293 cells assessed as stimulation of cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50557261(CHEMBL4749279)
Affinity DataEC50:  30nMAssay Description:Agonist activity at rat glucagon receptor expressed in HEK293 cells assessed as stimulation of cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50557262(CHEMBL4759334)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at rat glucagon receptor expressed in HEK293 cells assessed as stimulation of cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50557263(CHEMBL4752195)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at rat glucagon receptor expressed in HEK293 cells assessed as stimulation of cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50557264(CHEMBL4751466)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at rat glucagon receptor expressed in HEK293 cells assessed as stimulation of cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104037(His-Ser-Gln-Gly-Lys-Phe-Thr-Ser-Glu-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 0.200nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104040(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 0.240nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50122102(3-Cyano-4-hydroxy-benzoic acid [1-(2,3,5,6-tetrame...)
Affinity DataIC50: 0.430nMAssay Description:In vitro binding affinity towards rat glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50110054(3-Cyano-4-hydroxy-benzoic acid [1-[4-(4-isopropyl-...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibitory activity against rat glucagon receptor using [127I]-labeled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:Compound was tested for its ability to displace [125I]glucagon from the glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50051588(His-Ser-Gln-thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Tyr-Le...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098571(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 1.5nMAssay Description:In vitro receptor binding affinity (95% CL) using rat liver plasma membrane bioassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104030(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ly...)
Affinity DataIC50: 1.70nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50051586([des-His1,Tyr5,Glu9,D-Tyr10]glucagon-NH2 | CHEMBL4...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104039(His-Ser-Gln-Cys-Thr-Phe-Thr-Ser-Cys-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 3.60nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098563(Ser-Gln-Gly-Thr-Phe-Thr-Ser-Glu-Tyr-Ser-Lys-Tyr-Le...)
Affinity DataIC50: 3.75nMAssay Description:Compound was evaluated for its ability to displace radiolabeled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50407844(CHEMBL2115191)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50057796(CHEMBL3326188)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in rat hepatocytes after 15 mins by cAMP dynamic2 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/1/2016
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104031(His-Cys-Gln-Gly-Thr-Phe-Cys-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 5.60nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104043(His-Ser-Lys-Gly-Thr-Phe-Glu-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 6nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104041(His-Ser-Gln-Gly-Thr-Phe-Cys-Ser-Asp-Tyr-Ser-Cys-Ty...)
Affinity DataIC50: 6.40nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50454201(CHEMBL3037804)
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]glucagon binding towards Glucagon receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104033(His-Ser-Gln-Gly-Thr-Phe-Lys-Ser-Asp-Tyr-Glu-Lys-Ty...)
Affinity DataIC50: 14nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104044(His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Ty...)
Affinity DataIC50: 14nMAssay Description:Glucagon receptor binding measured as 50% inhibitory concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098573(N-trinitrophenyl-His-Ser-Gln-Gly-Thr-Phe-Thr-Ser-A...)
Affinity DataIC50: 15nMAssay Description:Compound was evaluated for its ability to displace radiolabeled glucagon (inactive up to 100 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50059352([des-His1, Trp6, Glu9] glucagon-NH2 | CHEMBL442499)
Affinity DataIC50: 19nMAssay Description:Binding affinity towards Glucagon receptor in rat liver plasma membranes by displacement of 125 I-labelled glucagonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098566(phenylbutyryl-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg-Arg-...)
Affinity DataIC50: 21.2nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50171817(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50: 23nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50104096(3-Chloro-4-hydroxy-benzoic acid (4-hydroxy-naphtha...)
Affinity DataIC50: 27nMAssay Description:Binding affinity towards rat Glucagon ReceptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50098572(Ac-Phe-Thr-Ser-Asp-Tyr-Ser-Lys-Tyr-Leu-Asp-Ser-Arg...)
Affinity DataIC50: 31nMAssay Description:IC50 value was expressed as inhibition of [125]glucagon specific binding.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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