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LigandPNGBDBM253928(US9464092, T | US9527857, T | US10189849, Compound...)
Affinity DataEC50: <100nMAssay Description:Inhibition of human CDK2/cyclin EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM253941(US9464092, GG | US9527857, GG)
Affinity DataEC50: <100nMAssay Description:Inhibition of human CDK2/cyclin EMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378288(CHEMBL567434)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378304(CHEMBL568080)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378305(CHEMBL583417)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378319(CHEMBL568303)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378289(CHEMBL565705)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378290(CHEMBL568310)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378291(CHEMBL568302)
Affinity DataIC50: 0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378292(CHEMBL566106)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50003691(CHEMBL567624)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378293(CHEMBL566550)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378294(CHEMBL566972)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378295(CHEMBL565490)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378298(CHEMBL583421)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378299(CHEMBL568079)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378297(CHEMBL566105)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378296(CHEMBL568510)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378301(CHEMBL568311)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378302(CHEMBL583615)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378300(CHEMBL565930)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378303(CHEMBL567208)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378212(CHEMBL575450)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378307(CHEMBL566329)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378312(CHEMBL578664)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378311(CHEMBL568301)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378308(CHEMBL568509)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378314(CHEMBL578256)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378310(CHEMBL566971)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378309(CHEMBL568093)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378313(CHEMBL567626)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50595815(CHEMBL5179962 | US11919904, Example 7)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged full-length CDK2/Flag-tagged cyclinE1 expressed in baculovirus expression system using eIF4E-bi...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50378315(CHEMBL578865)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378316(CHEMBL568291)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50595811(CHEMBL5194832)
Affinity DataIC50: 0.320nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged full-length CDK2/Flag-tagged cyclinE1 expressed in baculovirus expression system using eIF4E-bi...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50595809(CHEMBL5175160)
Affinity DataIC50: 0.330nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged full-length CDK2/Flag-tagged cyclinE1 expressed in baculovirus expression system using eIF4E-bi...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM601933(US11643416, Compound 1 | 4-((6'-hydroxy-8'-oxo-7',...)
Affinity DataIC50: 0.340nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, Calif.) to determine their inhibitory effect on these CDKs....More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM601933(US11643416, Compound 1 | 4-((6'-hydroxy-8'-oxo-7',...)
Affinity DataIC50: 0.340nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, CA) to determine their inhibitory effect on these CDKs. The...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM50378317(CHEMBL565273)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378318(CHEMBL566539)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM601934(US11643416, Compound 2 | 4-((7'-oxo-7',8'-dihydro-...)
Affinity DataIC50: 0.5nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, Calif.) to determine their inhibitory effect on these CDKs....More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM601934(US11643416, Compound 2 | 4-((7'-oxo-7',8'-dihydro-...)
Affinity DataIC50: 0.5nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, CA) to determine their inhibitory effect on these CDKs. The...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 0.520nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM601935(US11643416, Compound 3 | 4-((3'-oxo-2',3'-dihydro-...)
Affinity DataIC50: 0.560nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, Calif.) to determine their inhibitory effect on these CDKs....More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM601935(US11643416, Compound 3 | 4-((3'-oxo-2',3'-dihydro-...)
Affinity DataIC50: 0.560nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, CA) to determine their inhibitory effect on these CDKs. The...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM50595813(CHEMBL5190590 | US11919904, Example 15)
Affinity DataIC50: 0.620nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged full-length CDK2/Flag-tagged cyclinE1 expressed in baculovirus expression system using eIF4E-bi...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50511924(CHEMBL2377864)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of GST-tagged CDK2/Cyclin E (unknown origin) expressed in baculovirus expression system using GST-pRb (776 to 928 residues) as substrate m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase 3/G1/S-specific cyclin-E1(Human)
G1 Therapeutics

US Patent
LigandPNGBDBM601933(US11643416, Compound 1 | 4-((6'-hydroxy-8'-oxo-7',...)
Affinity DataIC50: 0.940nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, Calif.) to determine their inhibitory effect on these CDKs....More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetCyclin-dependent kinase 3/G1/S-specific cyclin-E1(Human)
G1 Therapeutics

US Patent
LigandPNGBDBM601933(US11643416, Compound 1 | 4-((6'-hydroxy-8'-oxo-7',...)
Affinity DataIC50: 0.940nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, CA) to determine their inhibitory effect on these CDKs. The...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM50378306(CHEMBL567647)
Affinity DataIC50: 0.950nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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