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TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50411311(CHEMBL2113267)
Affinity DataIC50: 1.30E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50292287(CHEMBL465161 | ginkgolide-A | GINKGOLIDE A)
Affinity DataIC50: 2.10E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50251276(CHEMBL514432 | BN 52021 | ginkgolide B | Gingkolid...)
Affinity DataIC50: 3.70E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208068((1R,3R,6R,7S,8S,9S,10R,11R,12R,13S,16S,17R)-8-tert...)
Affinity DataIC50: 4.60E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208060(10-methoxy-ginkgolide C | CHEMBL221823)
Affinity DataIC50: 7.80E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(ginkgolide C | CHEMBL221821)
Affinity DataIC50: 8.20E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208076(3,14-didehydroginkgolide A | CHEMBL373969)
Affinity DataIC50: 9.50E+3nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208074(ginkgolide J | CHEMBL374004)
Affinity DataIC50: 1.20E+4nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208085((3S,8R,12R,16S,17R,21S)-3-tert-butyl-17-hydroxy-16...)
Affinity DataIC50: 1.20E+4nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208081((1R,3R,6R,7S,8S,9S,10R,11R,12R,13S,16S,17R)-8-tert...)
Affinity DataIC50: 1.30E+4nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208082((1R,3R,6R,7S,8S,9S,10S,11R,12R,13S,16S,17R)-9-azid...)
Affinity DataIC50: 2.90E+4nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2/beta(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50459893(Gelsemine)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant human glycine receptor alpha2beta expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208091((1S,6R,8S,11R,12R,13S,16S,17R)-8-tert-butyl-6,12,1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208061((1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-tert-butyl-9-(...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208087(10-acetoxy-ginkgolide B | CHEMBL222222)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208079((1R,6R,8S,11R)-8-tert-butyl-13-methoxy-5,15,16-tri...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208090((1S,8S,11S,13S,16S,17R)-8-tert-butyl-17-hydroxy-16...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208069((1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-tert-butyl-6,1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208089((1R,6R,8S,11S,13S,16R,17R)-8-tert-butyl-16-methyl-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208080(1,2;3,14-dianhydro-ginkgolide C | CHEMBL412540)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208092((1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-tert-butyl-6,1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208083((1S,6R,8S,11S,13R,16R,17R)-8-tert-butyl-6,17-dihyd...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208065(methyl 2-[(1R,6R,8S,11S,14E)-8-tert-butyl-6-hydrox...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208067(methyl (2R)-2-[(1S,2R,3S,6S,8S,10S)-10-tert-butyl-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208072((1S,2R,3S,6S,8S,10R)-10-tert-butyl-2-hydroxy-3-met...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208086((1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-tert-butyl-6,1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208063(10-methoxymethyloxy-ginkgolide A | CHEMBL225470)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208088(methyl 2-[(1R,6R,8S,11S,14R)-8-tert-butyl-6-hydrox...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208059(CHEMBL412384)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208078((6R,8S,11S,16R,17S)-8-tert-butyl-6,16,17-trihydrox...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208077((1S,6R,8S,9R,11S,12R,13S,16S,17R)-8-tert-butyl-6,1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208075((1S,6R,8S,11S,13S,16R,17R)-8-tert-butyl-6,17-dihyd...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208070((1S,6R,8S,9S,11R,12R,13S,16S,17R)-8-tert-butyl-6,9...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208066((1R,2R,3S,6S,8S,10R,11R)-10-tert-butyl-2,11,16-tri...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycine receptor subunit alpha-2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208062((1R,6R,8S,11S)-8-tert-butyl-6,13-dimethoxy-2,4,14,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at human alpha-2GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed