Compile Data Set for Download or QSAR
Report error Found 78 of affinity data for UniProtKB/TrEMBL: P0DMV8
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM82124(adenosine-derived inhibitor (Grp78), 1)
Affinity DataKd:  500nMpH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA1A (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32381(adenosine-derived inhibitor (Grp78), 14 | adenosin...)
Affinity DataKd:  50nMpH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32378(adenosine-derived inhibitor (Grp78), 13 | adenosin...)
Affinity DataKd:  300nMpH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32370(adenosine-derived inhibitor (Grp78), 2 | adenosine...)
Affinity DataKd:  1.10E+4nMpH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM31995(ADP | CHEMBL14830 | Adenosine Diphosphate (ADP))
Affinity DataKd:  500nMpH: 7.4 T: 2°CAssay Description:All experiments were performed on a Biacore T100 at 25 deg C with a flow rate of 30 uL per minute. Double His-tagged HSP70 was immobilised on the sur...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32383(adenosine-derived inhibitor, 17)
Affinity DataKd:  120nMpH: 7.4 T: 2°CAssay Description:All experiments were performed on a Biacore T100 at 25 deg C with a flow rate of 30 uL per minute. Double His-tagged HSP70 was immobilised on the sur...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32382(adenosine-derived inhibitor, 16)
Affinity DataKd:  60nMpH: 7.4 T: 2°CAssay Description:All experiments were performed on a Biacore T100 at 25 deg C with a flow rate of 30 uL per minute. Double His-tagged HSP70 was immobilised on the sur...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32381(adenosine-derived inhibitor (Grp78), 14 | adenosin...)
Affinity DataKd:  50nMpH: 7.4 T: 2°CAssay Description:All experiments were performed on a Biacore T100 at 25 deg C with a flow rate of 30 uL per minute. Double His-tagged HSP70 was immobilised on the sur...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32380(adenosine-derived inhibitor, 14)
Affinity DataKd:  4.20E+3nMpH: 7.4 T: 2°CAssay Description:All experiments were performed on a Biacore T100 at 25 deg C with a flow rate of 30 uL per minute. Double His-tagged HSP70 was immobilised on the sur...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32379(adenosine-derived inhibitor, 13)
Affinity DataKd:  200nMpH: 7.4 T: 2°CAssay Description:All experiments were performed on a Biacore T100 at 25 deg C with a flow rate of 30 uL per minute. Double His-tagged HSP70 was immobilised on the sur...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32378(adenosine-derived inhibitor (Grp78), 13 | adenosin...)
Affinity DataKd:  300nMpH: 7.4 T: 2°CAssay Description:All experiments were performed on a Biacore T100 at 25 deg C with a flow rate of 30 uL per minute. Double His-tagged HSP70 was immobilised on the sur...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32370(adenosine-derived inhibitor (Grp78), 2 | adenosine...)
Affinity DataKd:  1.10E+4nMpH: 7.4 T: 2°CAssay Description:All experiments were performed on a Biacore T100 at 25 deg C with a flow rate of 30 uL per minute. Double His-tagged HSP70 was immobilised on the sur...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32383(adenosine-derived inhibitor, 17)
Affinity DataIC50: 400nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM31995(ADP | CHEMBL14830 | Adenosine Diphosphate (ADP))
Affinity DataIC50: 500nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM2(CHEMBL14249 | ({[({[(2R,3S,4R,5R)-5-(6-amino-9H-pu...)
Affinity DataIC50: 500nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32378(adenosine-derived inhibitor (Grp78), 13 | adenosin...)
Affinity DataIC50: 500nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32382(adenosine-derived inhibitor, 16)
Affinity DataIC50: 600nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32381(adenosine-derived inhibitor (Grp78), 14 | adenosin...)
Affinity DataIC50: 900nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32379(adenosine-derived inhibitor, 13)
Affinity DataIC50: 1.30E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32380(adenosine-derived inhibitor, 14)
Affinity DataIC50: 1.70E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32377(adenosine-derived inhibitor (Grp78), 12 | adenosin...)
Affinity DataIC50: 2.40E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32375(adenosine-derived inhibitor (Grp78), 9 | adenosine...)
Affinity DataIC50: 2.90E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32376(adenosine-derived inhibitor (Grp78), 11 | adenosin...)
Affinity DataIC50: 3.20E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32374(adenosine-derived inhibitor, 8)
Affinity DataIC50: 4.90E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32373(adenosine-derived inhibitor (Grp78), 8 | adenosine...)
Affinity DataIC50: 9.10E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32370(adenosine-derived inhibitor (Grp78), 2 | adenosine...)
Affinity DataIC50: 9.40E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32372(adenosine-derived inhibitor, 6)
Affinity DataIC50: 1.00E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM32371(adenosine-derived inhibitor (Grp78), 3 | adenosine...)
Affinity DataIC50: 1.70E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescein-labeled ATP-based probe was utilized, which binds to the GST fused ATPase domain (amino acids 3-383) of HSP70, producing an increase in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617260(CHEMBL5433282)
Affinity DataIC50: 2.52E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617272(CHEMBL5435048)
Affinity DataIC50: 4.73E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617266(CHEMBL5418499)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617288(CHEMBL5410116)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617267(CHEMBL5410567)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617268(CHEMBL5415571)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617269(CHEMBL5405780)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617270(CHEMBL5403880)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617271(CHEMBL5407447)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617273(CHEMBL5409255)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617274(CHEMBL5422252)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617275(CHEMBL5437667)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617263(CHEMBL5425589)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617276(CHEMBL5403845)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617277(CHEMBL5419391)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617278(CHEMBL5410605)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617279(CHEMBL5421614)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617280(CHEMBL5397525)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617281(CHEMBL5429240)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617282(CHEMBL5425293)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
Vernalis (R&D)

LigandPNGBDBM50617283(CHEMBL5395892)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA1A (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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