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TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM197051(US9212206, III)
Affinity DataIC50: 3.70nMpH: 7.4Assay Description:Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM197054(US9212206, VII)
Affinity DataIC50: 3.90nMpH: 7.4Assay Description:Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM197053(US9212206, VI)
Affinity DataIC50: 9.70nMpH: 7.4Assay Description:Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM197052(US9212206, V)
Affinity DataIC50: 26nMpH: 7.4Assay Description:Human aminopeptidase P2 (APP2) enzyme activity was determined using the internally quenched fluorescent substrate: H-Lys(2-aminobenzoyl)-Pro-Pro-p-ni...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078397(1-(3-Amino-2-hydroxy-5-methyl-hexanoyl)-pyrrolidin...)
Affinity DataIC50: 130nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078402((S)-1-((R)-3-Amino-2-hydroxy-5-methyl-hexanoyl)-py...)
Affinity DataIC50: 230nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078397(1-(3-Amino-2-hydroxy-5-methyl-hexanoyl)-pyrrolidin...)
Affinity DataIC50: 230nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078402((S)-1-((R)-3-Amino-2-hydroxy-5-methyl-hexanoyl)-py...)
Affinity DataIC50: 430nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078398(2-[(S)-2-((S)-1-Carbamoyl-ethylcarbamoyl)-pyrrolid...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078393((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078401((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078393((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078401((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078398(2-[(S)-2-((S)-1-Carbamoyl-ethylcarbamoyl)-pyrrolid...)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078391((S)-1-[(R)-3-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078391((S)-1-[(R)-3-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078392((S)-1-((2R,3R)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078392((S)-1-((2R,3R)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50351402(CHEMBL1819090)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078390((S)-1-((2S,3S)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078394((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078390((S)-1-((2S,3S)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078394((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078396((S)-1-(2-Mercapto-cyclopentanecarbonyl)-pyrrolidin...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078396((S)-1-(2-Mercapto-cyclopentanecarbonyl)-pyrrolidin...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078396((S)-1-(2-Mercapto-cyclopentanecarbonyl)-pyrrolidin...)
Affinity DataIC50: 3.90E+5nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078396((S)-1-(2-Mercapto-cyclopentanecarbonyl)-pyrrolidin...)
Affinity DataIC50: 3.90E+5nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078400(1-[1-(3-Amino-2-hydroxy-4-phenyl-butyryl)-4-hydrox...)
Affinity DataIC50: 4.70E+5nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078400(1-[1-(3-Amino-2-hydroxy-4-phenyl-butyryl)-4-hydrox...)
Affinity DataIC50: 6.00E+5nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078399((S)-1-((3R,4S)-4-Amino-3-hydroxy-6-methyl-heptanoy...)
Affinity DataIC50: 2.00E+6nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078399((S)-1-((3R,4S)-4-Amino-3-hydroxy-6-methyl-heptanoy...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetXaa-Pro aminopeptidase 2(Human)
TBA

US Patent
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed