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Report error Found 151 of affinity data for UniProtKB/TrEMBL: O43194
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030774(CHEMBL3342379)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030775(CHEMBL3342378)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030776(CHEMBL3342377)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030777(CHEMBL3342376)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030778(CHEMBL3342375)
Affinity DataEC50:  36nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030779(CHEMBL3342374)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030780(CHEMBL3342373)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030781(CHEMBL3342372)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030782(CHEMBL3342371)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030783(CHEMBL3342370)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030784(CHEMBL3342369)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030785(CHEMBL3342368)
Affinity DataEC50:  87nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030786(CHEMBL3342367)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030787(CHEMBL3342366)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030767(CHEMBL3342365)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030768(CHEMBL3342364)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030769(CHEMBL3342363)
Affinity DataEC50:  2.20E+4nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030770(CHEMBL3342362)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030771(CHEMBL3342361)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030772(CHEMBL3342360)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030773(CHEMBL3342359)
Affinity DataEC50:  164nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030788(CHEMBL3342358)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030788(CHEMBL3342358)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at human GPR39 by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030789(CHEMBL3341764)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR39 by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030790(CHEMBL3342357)
Affinity DataEC50:  202nMAssay Description:Agonist activity at human GPR39 by IP1 assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030788(CHEMBL3342358)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030777(CHEMBL3342376)
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030776(CHEMBL3342377)
Affinity DataEC50:  0.550nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50030774(CHEMBL3342379)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM16(zinc(2+) ion | Zn2+)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50044849(CHEMBL3311308)
Affinity DataEC50: <5.01E+4nMAssay Description:Agonist activity against human GPR39 expressed in CHO cells by BacMam IP1 HTRF/summary (Abse5) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50443616(CHEMBL3092413)
Affinity DataEC50:  900nMAssay Description:Agonist activity at GPR39 in human HT-29 cells assessed as increase in intracellular Ca2+ mobilization after 72 hrs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50443617(CHEMBL3092410)
Affinity DataEC50:  840nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced cAMP production preincubated for 30 mins m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50443618(CHEMBL3092411)
Affinity DataEC50:  310nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced cAMP production preincubated for 30 mins m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50443619(CHEMBL3092412)
Affinity DataEC50:  4.50E+3nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced cAMP production preincubated for 30 mins m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50443616(CHEMBL3092413)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced cAMP production preincubated for 30 mins m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50443617(CHEMBL3092410)
Affinity DataEC50:  190nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced intracellular Ca+2 mobilization after 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50443618(CHEMBL3092411)
Affinity DataEC50:  320nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced intracellular Ca+2 mobilization after 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50443619(CHEMBL3092412)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced intracellular Ca+2 mobilization after 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50443616(CHEMBL3092413)
Affinity DataEC50:  56nMAssay Description:Agonist activity at recombinant human GPR39 expressed in CHO-K1 cells assessed as increase of Zn2+-induced intracellular Ca+2 mobilization after 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50232365(CHEMBL4087979)
Affinity DataEC50:  388nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50232366(CHEMBL4065636)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50232367(CHEMBL4093273)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50232368(CHEMBL4095849)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50232369(CHEMBL4066831)
Affinity DataEC50:  460nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50232370(CHEMBL4060772)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation in presence of ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50232371(CHEMBL4099134)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation in presence of ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50232372(CHEMBL4063554)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation in presence of ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50232373(CHEMBL4101617)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation in presence of ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 39(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50232374(CHEMBL4083614)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GPR39 expressed in HEK293 cells co-expressing Galphaq assessed as myo-[2-3H]inositol phosphate accumulation in presence of ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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