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Report error Found 8 of affinity data for UniProtKB/TrEMBL: D3Z7P3
TargetGlutaminase kidney isoform, mitochondrial(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataIC50: 20nMAssay Description:Inhibition of GLS1 in mouse kidney assessed as inhibition of glutamate production using glutamine as substrate incubated for 1 hr by coupled assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataIC50: 20nMAssay Description:Inhibition of GLS1 in mouse brain assessed as inhibition of glutamate production using glutamine as substrate incubated for 1 hr by coupled assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503321(CHEMBL4540444)
Affinity DataIC50: 25nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation at 0.1 uM using glutamine as substrate by Nessler's reagent based assay relative...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503289(CHEMBL4462220)
Affinity DataIC50: 50nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation at 0.1 uM using glutamine as substrate by Nessler's reagent based assay relative...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503291(CHEMBL4562029)
Affinity DataIC50: 50nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation using glutamine as substrate by Nessler's reagent based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503294(CHEMBL4577734)
Affinity DataIC50: 50nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation at 0.1 uM using glutamine as substrate by Nessler's reagent based assay relative...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503296(CHEMBL4452754)
Affinity DataIC50: 50nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation at 0.1 uM using glutamine as substrate by Nessler's reagent based assay relative...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50503312(CHEMBL4537860)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse kidney glutaminase assessed as ammonia formation at 0.1 uM using glutamine as substrate by Nessler's reagent based assay relative...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed