Assay Method Information

Assay Name:  ChEMBL_1614374 (CHEMBL3856443)
Description:  Partial antagonist activity at rat TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced inward current at -60 mV holding potential pretreated for 180 secs prior to capsaicin addition in presence of extracellular calcium by whole-cell patch-clamp method
Affinity data for this assay
 

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