Assay Method Information

Assay Name:  ChEMBL_1838325 (CHEMBL4338458)
Description:  Inhibition of recombinant human C-terminal His-fusion tagged/N-terminal Strep-2 tagged HDAC8 (1 to 377 residues) expressed in insect cells using Boc-Lys(TFa)-AMC as substrate preincubated for 5 mins followed by substrate addition measured after 90 mins by fluorescence assay
Affinity data for this assay
 

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