Assay Method Information

Assay Name:  ChEMBL_1724088 (CHEMBL4139366)
Description:  Antagonist activity at human vasopressin 1a receptor expressed in HEK293 cell membranes assessed as inhibition of AVP-induced increase in Ca2+ flux preincubated for 5 mins followed by AVP addition measured after 5 mins for every 2 secs by Ca5 dye based FLIPR assay
Affinity data for this assay
 

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