Assay Method Information

Assay Name:  ChEMBL_2057194 (CHEMBL4712195)
Description:  Antagonist activity at human C-terminal GFP10-fused GPR84 expressed in HEK293 cells co-expressing Rluc8-tagged Galphai2/GFP10-tagged Ggamma2/Gbeta1 assessed as inhibition of embelin-induced Galphai activation incubated for 10 mins by BRET assay
Affinity data for this assay
 

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