| Assay Method Information | |
| | ChEMBL_2056372 (CHEMBL4711373) |
| Description: | Non-competitive antagonist activity at human CB2R expressed in CHO cell membranes assessed as N-cycloheptyl-1,2-dihydro-1-(4-fluorobenzyl)-6-methyl-2-oxo-5-phenyl-pyridine-3-carboxamide EC50 at 1000 nM preincubated with compound for 30 mins followed by GTPgammaS addition and measured after 90 mins by [35S]GTPgammaS assay (Rvb = 19.4 nM) |
| Affinity data for this assay | |
|---|---|
| If you find an error in this entry please send us an E-mail | |