| Assay Method Information | |
| | ChEMBL_2056369 (CHEMBL4711370) |
| Description: | Competitive antagonist activity at human CB2R expressed in CHO cell membranes assessed as rightward shift of N-cycloheptyl-1,2-dihydro-5-bromo-1-(4-fluoro benzyl)-6-methyl-2-oxo-pyridine-3-carboxamide-induced GTPgammaS binding by measuring N-cycloheptyl-1,2-dihydro-5-bromo-1-(4-fluoro benzyl)-6-methyl-2-oxo-pyridine-3-carboxamide EC50 at 1000 nM preincubated with compound for 30 mins followed by GTPgammaS addition and measured after 90 mins by [35S]GTPgammaS assay (Rvb = 11.6 nM) |
| Affinity data for this assay | |
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