Assay Method Information

Assay Name:  ChEMBL_815799 (CHEMBL2025966)
Description:  Antagonist activity at human alpha4beta2 nAChR expressed in SH-EP1 cells assessed as inhibition of carbamylcholine induced 86Rb+ ion efflux preincubated for 10 mins prior to carbamylcholine-induction measured after 5 mins by flip-plate technique
Affinity data for this assay
 

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