| Assay Method Information | |
| | ChEMBL_1927520 (CHEMBL4430592) |
| Description: | Antagonist activity against human GnRH receptor expressed in HEK293 cells co-transfected with pGL4-NFAT promoter AP1-luc assessed as inhibition of 20 nM GnRH-induced NFAT activation pre-incubated for 1 hr before GnRH stimulation and measured after 6 hrs by luciferase reporter gene assay |
| Affinity data for this assay | |
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