Assay Method Information

Assay Name:  ChEMBL_1889207 (CHEMBL4390961)
Description:  Agonist activity at human mu opioid receptor expressed in CHOK1 cells coexpressing Galpha15 assessed as increase in intracellular calcium flux in presence of mu opioid receptor antagonist naloxone and incubated for 1 hr measured for 90 secs at 1.5 sec interval by FLIPR assay
Affinity data for this assay
 

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