| Assay Method Information | |
| | ChEMBL_1721241 (CHEMBL4136241) |
| Description: | Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) Y537S mutant expressed in Escherichia coli assessed as inhibition of estradiol-induced fluorescein-labeled PGC1alpha coactivator peptide binding after overnight incubation by Lantascreen TR-FRET assay |
| Affinity data for this assay | |
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