Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 4222
LigandPNGBDBM54950(6-cyclohexyl-3-(2-furanyl)-[1,2,4]triazolo[3,4-b][...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM38325(cid_662931 | 6-(3,4-dimethoxyphenyl)-3-(2-pyridiny...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54951((6Z)-3-(2-furanyl)-6-(2-pyrrolylidene)-5H-[1,2,4]t...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54952(6-cycloheptyl-3-(2-furanyl)-[1,2,4]triazolo[3,4-b]...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54953(3-(2-furanyl)-6-(2-methoxy-4-nitrophenyl)-[1,2,4]t...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54954(VU0364704-1 | 6-cyclohexyl-3-pyridin-2-yl-[1,2,4]t...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54955(cid_44236877 | (6Z)-3-(2-pyridinyl)-6-(2-pyrrolyli...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54956(cid_44236878 | 6-cycloheptyl-3-pyridin-2-yl-[1,2,4...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54957(cid_44236879 | 6-(2-methoxy-4-nitrophenyl)-3-pyrid...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54958(cid_662681 | 6-(3-methoxyphenyl)-3-(2-pyridinyl)-[...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54959(6-(3-ethoxyphenyl)-3-(2-furanyl)-[1,2,4]triazolo[3...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54960(cid_663172 | VU0247748-2 | 3-pyridin-4-yl-6-(thiop...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54961(6-(3-ethoxyphenyl)-3-thiophen-2-yl-[1,2,4]triazolo...)
Affinity DataEC50: >3.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay