Compile Data Set for Download or QSAR
Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 3284
TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110971(US8614253, 3-2 | US9241942, 3-2 | US9963434, Compo...)
Affinity DataIC50: 30nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110970(US8614253, 3-1 | US9241942, 3-1 | US9963434, Compo...)
Affinity DataIC50: 30nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110972(US8614253, 43-10 | US8614253, 3-3 | US9241942, 3-3...)
Affinity DataIC50: 40nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110973(US8614253, 43-81 | US8614253, 3-4 | US9241942, 3-4...)
Affinity DataIC50: 70nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110974(US8614253, 3-5 | US9241942, 3-5 | US9963434, Compo...)
Affinity DataIC50: 80nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110975(US8614253, 43-4 | US8614253, 3-6 | US9241942, 3-6 ...)
Affinity DataIC50: 100nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110976(US8614253, 3-7 | US9241942, 3-7 | US9963434, Compo...)
Affinity DataIC50: 110nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM202537(US9241942, 3-8 | US9963434, Compound 3-8)
Affinity DataIC50: 120nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110978(US8614253, 3-9 | US9241942, 3-9 | US9963434, Compo...)
Affinity DataIC50: 170nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110979(US8614253, 42-1 | US8614253, 43-1 | US8614253, 3-1...)
Affinity DataIC50: 170nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110980(US8614253, 3-11 | US9241942, 3-11 | US9963434, Com...)
Affinity DataIC50: 240nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110981(US8614253, 3-12 | US9241942, 3-12 | US9963434, Com...)
Affinity DataIC50: 240nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110982(US8614253, 3-13 | US9241942, 3-13 | US9963434, Com...)
Affinity DataIC50: 250nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110983(US8614253, 43-5 | US8614253, 42-12 | US8614253, 3-...)
Affinity DataIC50: 270nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110984(US8614253, 3-15 | US9241942, 3-15 | US9963434, Com...)
Affinity DataIC50: 280nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110985(US8614253, 26-2 | US8614253, 3-16 | US9241942, 3-1...)
Affinity DataIC50: 300nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110986(US8614253, 3-17 | US9241942, 3-17 | US9963434, Com...)
Affinity DataIC50: 350nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110987(US8614253, 3-18 | US9241942, 3-18 | US9963434, Com...)
Affinity DataIC50: 380nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110988(US8614253, 3-19 | US9241942, 3-19 | US9963434, Com...)
Affinity DataIC50: 380nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110989(US8614253, 3-20 | US9241942, 3-20 | US9963434, Com...)
Affinity DataIC50: 390nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110990(US8614253, 3-21 | US9241942, 3-21 | US9963434, Com...)
Affinity DataIC50: 400nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110992(US8614253, 3-23 | US9241942, 3-23 | US9963434, Com...)
Affinity DataIC50: 400nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110991(US8614253, 3-22 | US9241942, 3-22 | US9963434, Com...)
Affinity DataIC50: 400nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110993(US8614253, 43-2 | US8614253, 3-24 | US9241942, 3-2...)
Affinity DataIC50: 410nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110994(US8614253, 3-25 | US9241942, 3-25 | US9963434, Com...)
Affinity DataIC50: 440nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110995(US8614253, 3-26 | US9241942, 3-26 | US9963434, Com...)
Affinity DataIC50: 510nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110996(US8614253, 3-27 | US9241942, 3-27 | US9963434, Com...)
Affinity DataIC50: 540nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110997(US8614253, 3-28 | US9241942, 3-28 | US9963434, Com...)
Affinity DataIC50: 550nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110998(US8614253, 3-29 | US9241942, 3-29 | US9963434, Com...)
Affinity DataIC50: 570nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM110999(US8614253, 26-1 | US8614253, 3-30 | US9241942, 3-3...)
Affinity DataIC50: 580nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111000(US8614253, 3-31 | US9241942, 3-31 | US9963434, Com...)
Affinity DataIC50: 720nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111001(US8614253, 3-32 | US9241942, 3-32 | US9963434, Com...)
Affinity DataIC50: 750nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111002(US8614253, 3-33 | US9241942, 3-33 | US9963434, Com...)
Affinity DataIC50: 750nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111003(US8614253, 3-34 | US9241942, 3-34 | US9963434, Com...)
Affinity DataIC50: 790nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111004(US8614253, 3-35 | US9241942, 3-35 | US9963434, Com...)
Affinity DataIC50: 990nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111005(US8614253, 3-36 | US9241942, 3-36 | US9963434, Com...)
Affinity DataIC50: 1.01E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111006(US8614253, 3-37 | US9241942, 3-37 | US9963434, Com...)
Affinity DataIC50: 1.07E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111007(US8614253, 3-38 | US9241942, 3-38 | US9963434, Com...)
Affinity DataIC50: 1.10E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111009(US8614253, 3-40 | US9241942, 3-40 | US9963434, Com...)
Affinity DataIC50: 1.28E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111008(US8614253, 3-39 | US9241942, 3-39 | US9963434, Com...)
Affinity DataIC50: 1.28E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111011(US8614253, 3-42 | US9241942, 3-42 | US9963434, Com...)
Affinity DataIC50: 1.30E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111010(US8614253, 3-41 | US9241942, 3-41 | US9963434, Com...)
Affinity DataIC50: 1.30E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111012(US8614253, 3-43 | US9241942, 3-43 | US9963434, Com...)
Affinity DataIC50: 1.31E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111013(US8614253, 3-44 | US9241942, 3-44 | US9963434, Com...)
Affinity DataIC50: 1.33E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111014(US8614253, 3-45 | US9241942, 3-45 | US9963434, Com...)
Affinity DataIC50: 1.38E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111015(US8614253, 3-46 | US9241942, 3-46 | US9963434, Com...)
Affinity DataIC50: 1.40E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111016(US8614253, 3-47 | US9241942, 3-47 | US9963434, Com...)
Affinity DataIC50: 1.48E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
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TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111017(US8614253, 3-48 | US9241942, 3-48 | US9963434, Com...)
Affinity DataIC50: 1.59E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111018(US8614253, 3-49 | US9241942, 3-49 | US9963434, Com...)
Affinity DataIC50: 1.64E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase/endoribonuclease IRE1(Human)
Fosun Orinove Pharmatech

US Patent
LigandPNGBDBM111019(US8614253, 3-50 | US9241942, 3-50 | US9963434, Com...)
Affinity DataIC50: 1.75E+3nMAssay Description:A fusion protein comprising glutathione S transferase (GST) and human IRE-1α (GST-IRE-1α) was obtained from a 500 ml baculovirus-infected i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2020
Entry Details
Go to US Patent

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