Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 3184
TargetP2X purinoceptor 4(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM393615(US09969700, 173)
Affinity DataIC50: 64nMAssay Description:The P2X4 receptor antagonist activity of the compounds of the present invention was measured as follows. The 1321N1 cells stably expressing human P2X...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2020
Entry Details
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TargetP2X purinoceptor 4(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM393614(US09969700, 48)
Affinity DataIC50: 430nMAssay Description:The P2X4 receptor antagonist activity of the compounds of the present invention was measured as follows. The 1321N1 cells stably expressing human P2X...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2020
Entry Details
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TargetP2X purinoceptor 4(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM393617(US09969700, 197)
Affinity DataIC50: 440nMAssay Description:The P2X4 receptor antagonist activity of the compounds of the present invention was measured as follows. The 1321N1 cells stably expressing human P2X...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2020
Entry Details
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TargetP2X purinoceptor 4(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM393612(US09969700, 13 | 5-[4-[(2-Chlorophenylacetyl)amino...)
Affinity DataIC50: 540nMAssay Description:The P2X4 receptor antagonist activity of the compounds of the present invention was measured as follows. The 1321N1 cells stably expressing human P2X...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2020
Entry Details
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TargetP2X purinoceptor 4(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM393616(US09969700, 196)
Affinity DataIC50: 970nMAssay Description:The P2X4 receptor antagonist activity of the compounds of the present invention was measured as follows. The 1321N1 cells stably expressing human P2X...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2020
Entry Details
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TargetP2X purinoceptor 4(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM393613(US09969700, 20)
Affinity DataIC50: 1.20E+3nMAssay Description:The P2X4 receptor antagonist activity of the compounds of the present invention was measured as follows. The 1321N1 cells stably expressing human P2X...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2020
Entry Details
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TargetP2X purinoceptor 4(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM393619(US09969700, 106 | 5-[4-(2-Iodobenzoyl)aminophenyl]...)
Affinity DataIC50: 1.80E+3nMAssay Description:The P2X4 receptor antagonist activity of the compounds of the present invention was measured as follows. The 1321N1 cells stably expressing human P2X...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2020
Entry Details
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TargetP2X purinoceptor 4(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM22416(PAROXETINE | CHEMBL490 | (3S,4R)-3-[(1,3-benzodiox...)
Affinity DataIC50: 4.00E+3nMAssay Description:The P2X4 receptor antagonist activity of the compounds of the present invention was measured as follows. The 1321N1 cells stably expressing human P2X...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/6/2020
Entry Details
Go to US Patent