Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 3016
TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388463(US9944606, Compound 701 | (1aS,5aS)-2-(4-Oxy-pyraz...)
Affinity DataKi:  1.45nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2020
Entry Details
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TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388466(US9944606, Compound 755 | (1aR,5aR)-2-(4-Oxy-pyraz...)
Affinity DataKi:  3.80nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2020
Entry Details
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TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388465(US9944606, Compound 752 | (1aR,5aR)-2-(Tetrahydro-...)
Affinity DataKi:  58.7nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388461(US9944606, Compound 64 | (1aS,5aS)-2-(2,4-Difluoro...)
Affinity DataKi:  97.6nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388462(US9944606, Compound 629 | (1aR,5aR)-2-(4-Oxy-pyraz...)
Affinity DataKi:  97.7nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388463(US9944606, Compound 701 | (1aS,5aS)-2-(4-Oxy-pyraz...)
Affinity DataKi:  105nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388461(US9944606, Compound 64 | (1aS,5aS)-2-(2,4-Difluoro...)
Affinity DataKi:  207nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388465(US9944606, Compound 752 | (1aR,5aR)-2-(Tetrahydro-...)
Affinity DataKi:  568nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Human)
Arena Pharmaceuticals

US Patent
LigandPNGBDBM388466(US9944606, Compound 755 | (1aR,5aR)-2-(4-Oxy-pyraz...)
Affinity DataKi:  1.20E+3nMAssay Description:Preparation of Membranes: HEK293 cells stably expressing human CB2 receptor were collected, washed in ice cold PBS, and centrifuged at 48,000×g for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2020
Entry Details
Go to US Patent