Compile Data Set for Download or QSAR
Report error Found 196 Enz. Inhib. hit(s) with all data for entry = 2675
TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344018(US9777017, Example 10 | US9777017, Example 2 | US9...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344020(US9777017, Example 4 | US9908895, Example 4 | US10...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344021(US9777017, Example 5 | US9908895, Example 5 | US10...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344023(US9777017, Example 7 | US9908895, Example 7 | US10...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344024(US9777017, Example 8 | US9908895, Example 8 | US10...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344018(US9777017, Example 10 | US9777017, Example 2 | US9...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344027(US9777017, Example 11 | US9908895, Example 11 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344028(US9777017, Example 12 | US9908895, Example 12 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344029(US9777017, Example 13 | US9908895, Example 13 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344033(US9777017, Example 17 | US9908895, Example 17 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344034(US9777017, Example 18 | US9908895, Example 18 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM246852(((2R,5S)-5-{2-[(1R)- 1-hydroxyethyl]-1H- imidazo[4...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344018(US9777017, Example 10 | US9777017, Example 2 | US9...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344040(US9777017, Example 24 | US9908895, Example 24 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344041(US9777017, Example 25 | US9908895, Example 25 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344042(US9777017, Example 26 | US9908895, Example 26 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344043(US9777017, Example 27 | US9908895, Example 27 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344048(US9777017, Example 32 | US9908895, Example 32 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344049(US9777017, Example 33 | US9908895, Example 33 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344051(US9777017, Example 35 | US9908895, Example 35 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344052(US9777017, Example 36 | US9908895, Example 36 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344052(US9777017, Example 36 | US9908895, Example 36 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344053(US9777017, Example 37 | US9908895, Example 37 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK1(Human)
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LigandPNGBDBM344054(US9777017, Example 38 | US9908895, Example 38 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
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TargetTyrosine-protein kinase JAK2(Human)
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US Patent
LigandPNGBDBM344054(US9777017, Example 38 | US9908895, Example 38 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344055(US9777017, Example 39 | US9908895, Example 39 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM375666(US9908895, Example 40 | US9908895, Example 41 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM375666(US9908895, Example 40 | US9908895, Example 41 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344058(US9777017, Example 42 | US9908895, Example 42 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344059(US9777017, Example 43 | US9908895, Example 43 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344061(US9777017, Example 45 | US9908895, Example 45 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344062(US9777017, Example 46 | US9908895, Example 46)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344063(US9777017, Example 47 | US9908895, Example 47 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344064(US9777017, Example 48 | US9908895, Example 48 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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US Patent
LigandPNGBDBM344064(US9777017, Example 48 | US9908895, Example 48 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344073(US9777017, Example 57 | US9908895, Example 57 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344074(US9777017, Example 58 | US9908895, Example 58 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344080(US9777017, Example 64 | US9908895, Example 64 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM375694(US9908895, Example 68)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344087(US9777017, Example 71 | US9908895, Example 71 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344088(US9777017, Example 72 | US9908895, Example 72 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344089(US9777017, Example 73 | US9908895, Example 73 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344091(US9777017, Example 75 | US9908895, Example 75 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344092(US9777017, Example 76 | US9908895, Example 76 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344093(US9777017, Example 77 | US9908895, Example 77 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
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US Patent
LigandPNGBDBM344093(US9777017, Example 77 | US9908895, Example 77 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344094(US9777017, Example 78 | US9908895, Example 78 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344095(US9777017, Example 79 | US9908895, Example 79 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344096(US9777017, Example 80 | US9908895, Example 80 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
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Date in BDB:
1/27/2020
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
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US Patent
LigandPNGBDBM344097(US9777017, Example 81 | US9908895, Example 81 | US...)
Affinity DataIC50: 100nMAssay Description:Compounds herein were tested for inhibitory activity of JAK targets according to the following in vitro assay described in Park et al., Analytical Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details
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